SCHEMBL9757026

SCHEMBL9757026

Cc1c(C(=O)O)sc2ccc(CBr)cc12

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 4/20 0.58
GPR35 Q9HC97 4/20 0.54
RXFP1 Q9HBX9 3/20 0.44
PKM P14618 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
PRNP P04156 1/20 0.41
MCL1 Q07820 4/20 0.40
BCL2L1 Q07817 2/20 0.40
HSD11B1 P28845 1/20 0.38
EDNRA P25101 1/20 0.38
ROCK1 Q13464 1/20 0.37
BCKDK O14874 1/20 0.36
CYP4F2 P78329 1/20 0.35
CYP4A11 Q02928 1/20 0.35
BCL2 P10415 1/20 0.35
BAD Q92934 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31207832 0.88 TBXAS1 (0.58) TBXAS1GPR35RXFP1PKMNPSR1
SCHEMBL10948748 0.86 TBXAS1 (0.60) TBXAS1GPR35RXFP1PKMNPSR1
SCHEMBL9613211 0.86 TBXAS1 (0.60) TBXAS1GPR35RXFP1PKMNPSR1
SCHEMBL2896475 0.80 GPR35 (0.58) TBXAS1GPR35RXFP1PKMNPSR1
SCHEMBL2895952 0.79 GPR35 (0.62) TBXAS1GPR35RXFP1PKMNPSR1
SCHEMBL9757077 0.78 GPR35 (0.65) TBXAS1GPR35RXFP1PKMNPSR1
SCHEMBL1066852 0.76 GPR35 (0.58) TBXAS1GPR35RXFP1PKMNPSR1
SCHEMBL122587 0.76 GPR35 (0.58) TBXAS1GPR35RXFP1PKMNPSR1
SCHEMBL2893771 0.76 GPR35 (0.58) TBXAS1GPR35RXFP1PKMNPSR1
SCHEMBL11287291 0.75 TBXAS1 (0.55) TBXAS1GPR35RXFP1PKMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019475-A2 QUINOLINYL-BENZOHETEROBICYCLIC DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D¿4? RHONE-POULENC RORER INTERNATIONAL (HOLDINGS) INC. (US) 1991-12-26 WO disclosed
US-5041453-A Quinolinyl-benzoheterobicyclic derivatives as antagonists of leukotriene D4 RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed