SCHEMBL11289658

SCHEMBL11289658

O=C(O)Oc1cc2c(s1)CCCNC2

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PNMT P11086 4/20 0.47
ITGB3 P05106 6/20 0.43
ITGA2B P08514 6/20 0.43
ALDH1A1 P00352 3/20 0.38
DAO P14920 1/20 0.38
TPSAB1 Q15661 1/20 0.36
TPSD1 Q9BZJ3 1/20 0.36
TPSG1 Q9NRR2 1/20 0.36
POLB P06746 2/20 0.35
PKM P14618 1/20 0.34
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33
PARP1 P09874 1/20 0.33
PARP2 Q9UGN5 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16712277 0.82 ALDH1A1 (0.56) ALDH1A1DAOPOLBPKMTP53
SCHEMBL16712269 0.82 DAO (0.56) ALDH1A1DAOPOLBPKMTP53
SCHEMBL1444085 0.79 PNMT (0.61) PNMTITGB3ITGA2BTPSAB1TPSD1
SCHEMBL6421249 0.78 ALDH1A1 (0.65) PNMTITGB3ITGA2BALDH1A1DAO
Hydrochloric Acid SCHEMBL1443367 0.78 PNMT (0.60) PNMTITGB3ITGA2BTPSAB1TPSD1
SCHEMBL15071934 0.75 PNMT (0.54) PNMTITGB3ITGA2BTPSAB1TPSD1
SCHEMBL18822929 0.75 PNMT (0.54) PNMTITGB3ITGA2BTPSAB1TPSD1
SCHEMBL9471965 0.75 PNMT (0.54) PNMTITGB3ITGA2BALDH1A1TPSAB1
Hydrochloric Acid SCHEMBL14141606 0.74 PNMT (0.52) PNMTITGB3ITGA2BTPSAB1TPSD1
SCHEMBL4397849 0.72 PNMT (0.61) PNMTITGB3ITGA2BTPSAB1TPSD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0058341-A1 Azepine derivatives, their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1982-08-25 EP disclosed