SCHEMBL11291680

SCHEMBL11291680

NCC(O)C1=CC2(CC2)c2ccccc21

nearest known ligand 0.33

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.33
TAAR1 Q96RJ0 2/20 0.31
HTR3A P46098 1/20 0.31
TSHR P16473 1/20 0.31
NFKB1 P19838 1/20 0.31
HIF1A Q16665 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALOX15 P16050 1/20 0.30
APEX1 P27695 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11290081 0.94 IDO1 (0.32) IDO1
SCHEMBL11294673 0.92 SLC6A4 (0.34) IDO1
SCHEMBL11291041 0.79 IDO1 (0.34) IDO1TAAR1HTR3ATSHRNFKB1
SCHEMBL11295572 0.78 LMNA (0.37)
SCHEMBL11289410 0.78
SCHEMBL31452460 0.75 SLC6A4 (0.34) TAAR1TSHRNFKB1HIF1AKDM4E
SCHEMBL11288858 0.75 SLC6A4 (0.34) TAAR1TSHRNFKB1HIF1AKDM4E
SCHEMBL11290059 0.75 RIPK1 (0.30)
SCHEMBL11290458 0.75 APOBEC3A (0.39)
SCHEMBL11349725 0.74 ADRB2 (0.41) TSHRNFKB1HIF1AKDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0000825-B1 GEMINALLY DISUBSTITUTED INDENE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Kabi AB (SE) 1982-04-14 EP disclosed
US-4218472-A USED AS DECONGESANT, HYPOTENSIVE AGENT, VASOCONSTRICTOR, ANTI-RESERPINE AGENT, TREATING INCONTINENCE AB KABI (SE) 1980-08-19 US disclosed
EP-0000825-A1 Geminally disubstituted indene derivatives, processes for their preparation and pharmaceutical compositions containing them Kabi AB (SE) 1979-02-21 EP disclosed