SCHEMBL1129302

SCHEMBL1129302

CC(C)(Cl)c1nc2cccc(F)c2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.37
NPSR1 Q6W5P4 1/20 0.35
CA12 O43570 1/20 0.35
CA9 Q16790 1/20 0.35
TNKS O95271 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35
PKM P14618 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
DAO P14920 1/20 0.32
DDO Q99489 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
PTGES O14684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22648457 0.86 PARP1 (0.39) PARP1NPSR1CA12CA9TNKS
SCHEMBL38663020 0.83 SCN10A (0.43) PARP1NPSR1CA12CA9TNKS
SCHEMBL1128774 0.81 NPSR1 (0.37) PARP1NPSR1NPC1RAB9AALDH1A1
SCHEMBL1128993 0.75 GAA (0.45) PARP1NPSR1TNKSTNKS2L3MBTL1
SCHEMBL5142221 0.73 PARP1 (0.59) PARP1CA12CA9TNKS2PKM
SCHEMBL9305632 0.73 CA12 (0.40) PARP1CA12CA9PKMNPC1
SCHEMBL23278130 0.72 CA12 (0.42) PARP1CA12CA9PKMNPC1
SCHEMBL20683086 0.70 SMN1; SMN2 (0.43) PARP1NPSR1CA12CA9PKM
SCHEMBL5508549 0.70 MEN1 (0.40) PARP1NPSR1NPC1RAB9AALDH1A1
SCHEMBL31741632 0.70 KDM4E (0.45) PARP1CA12CA9TNKSTNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2282762-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION Intermune, Inc. (US) 2011-02-16 EP disclosed
WO-2009142842-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2009-11-26 WO disclosed