Bicarbonate

Bicarbonate

SCHEMBL11298239

COc1ccc(CSc2nc(C)cc(C)n2)cc1.O=C(O)O

nearest known ligand 0.60

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.60
MIF P14174 1/20 0.60
HTT P42858 3/20 0.57
LMNA P02545 3/20 0.56
MMP13 P45452 1/20 0.56
SMN1; SMN2 Q16637 5/20 0.56
ALDH1A1 P00352 5/20 0.56
MAPT P10636 4/20 0.56
TDP1 Q9NUW8 3/20 0.56
RAB9A P51151 2/20 0.56
KMT2A Q03164 2/20 0.56
POLB P06746 2/20 0.56
MEN1 O00255 1/20 0.56
MITF O75030 1/20 0.56
PKM P14618 1/20 0.56
CTSB P07858 1/20 0.53
VCP P55072 1/20 0.53
L3MBTL1 Q9Y468 2/20 0.52
NPC1 O15118 1/20 0.52
TP53 P04637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16743643 0.86 HTT (0.54) KDM4EMIFHTTLMNAMMP13
SCHEMBL97659 0.79 NPC1 (0.54) KDM4ELMNAMMP13SMN1; SMN2ALDH1A1
SCHEMBL10691068 0.77 NPC1 (0.55) KDM4EHTTLMNAMMP13SMN1; SMN2
SCHEMBL14028274 0.77 HTT (0.60) KDM4EHTTLMNAMMP13SMN1; SMN2
SCHEMBL29935019 0.77 SMN1; SMN2 (0.57) HTTLMNAMMP13SMN1; SMN2ALDH1A1
SCHEMBL99151 0.76 NPC1 (0.54) KDM4ELMNAMMP13SMN1; SMN2ALDH1A1
SCHEMBL10913886 0.76 KDM4E (0.50) KDM4EMIFHTTSMN1; SMN2ALDH1A1
SCHEMBL5521119 0.75 MAOB (0.45) KDM4EMIFHTTLMNAMMP13
SCHEMBL10411023 0.73 HTT (0.70) KDM4EHTTLMNASMN1; SMN2ALDH1A1
SCHEMBL6637213 0.73 TP53 (0.56) KDM4ELMNAMMP13SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4337335-A Transition metal salt complexes of polyamino organic compounds SCHERING CORPORATION (US) 1982-06-29 US disclosed
US-4230847-A Aminoglycoside antibiotic compounds SCHERING CORPORATION (US) 1980-10-28 US disclosed