SCHEMBL11298796

SCHEMBL11298796

Cc1ccc(/N=c2\s[nH]c(=O)n2C2(c3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.36
CDC25A P30304 2/20 0.34
CDC25B P30305 2/20 0.34
MAPT P10636 4/20 0.34
KMT2A Q03164 4/20 0.34
MEN1 O00255 3/20 0.34
NPC1 O15118 3/20 0.34
RAB9A P51151 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LMNA P02545 2/20 0.32
AGTR1 P30556 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
MAPK1 P28482 1/20 0.31
MGAT2 Q10469 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18950494 0.94 CDC25A (0.37) CDC25ACDC25BMAPTKMT2AMEN1
SCHEMBL1047701 0.94 CDC25A (0.37) CDC25ACDC25BMAPTKMT2AMEN1
SCHEMBL1047702 0.94 CDC25A (0.37) CDC25ACDC25BMAPTKMT2AMEN1
SCHEMBL11298571 0.61 CCR2 (0.39) MAPTKMT2AMEN1NPSR1LMNA
SCHEMBL1051909 0.59 SMN1; SMN2 (0.38) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL18950440 0.59 SMN1; SMN2 (0.38) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL1051908 0.59 SMN1; SMN2 (0.38) MAPTKMT2AMEN1LMNAALDH1A1
SCHEMBL10813710 0.56 MAPT (0.52) MAPTKMT2AMEN1NPC1RAB9A
SCHEMBL73932 0.56 SLC6A4 (0.34) KMT2AMAPK1
SCHEMBL12346688 0.56 OPRM1 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9675596-B2 1,2,4-thiazolidin-3-one derivatives and their use in the treatment of cancer BALTIC BIO AB (SE) 2017-06-13 US disclosed
US-20160128993-A1 1,2,4-THIAZOLIDIN-3-ONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CANCER BALTICGRUPPEN BIO AB (SE) 2016-05-12 US disclosed
US-9162994-B2 1,2,4-thiazoloidin-3-one derivatives and their use in the treatment of cancer BETAGENON AB (SE) 2015-10-20 US disclosed
US-20120183537-A1 1,2,4-THIAZOLOIDIN-3-ONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CANCER BETAGENON AB 2012-07-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160128993-A1 1,2,4-THIAZOLIDIN-3-ONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CANCER HCCS, CCND3, MTNR1A HPGD 1539/4885CDC25A 366/4885CDC25B 438/4885
US-20120183537-A1 1,2,4-THIAZOLOIDIN-3-ONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF CANCER HCCS, CCND3, MTNR1A HPGD 1559/4885CDC25A 260/4885CDC25B 356/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.