SCHEMBL1129893

SCHEMBL1129893

CCc1nccc(-c2cc(=O)[nH]cn2)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.34
PARP1 P09874 6/20 0.33
ABL1 P00519 1/20 0.33
RIN1 Q13671 1/20 0.33
ACVR1 Q04771 1/20 0.33
PDE3B Q13370 2/20 0.32
PDE3A Q14432 2/20 0.32
CYP1A2 P05177 1/20 0.31
TMIGD3 P0DMS9 1/20 0.31
CYP2C9 P11712 1/20 0.31
ADORA1 P30542 1/20 0.31
IP6K1 Q92551 1/20 0.31
TBK1 Q9UHD2 1/20 0.31
KDM4A O75164 1/20 0.31
KDM4B O94953 1/20 0.31
KDM5C P41229 1/20 0.31
KDM5B Q9UGL1 1/20 0.31
GSK3B P49841 1/20 0.31
SLC2A1 P11166 1/20 0.31
CHEK1 O14757 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3825889 0.80 KDM4E (0.41) PARP1ABL1RIN1GSK3BCHEK1
SCHEMBL1129988 0.69 GRM5 (0.41) PARP1ABL1RIN1ADORA1IP6K1
SCHEMBL83683 0.67 KDM4E (0.52) SMN1; SMN2ABL1RIN1CYP1A2IP6K1
SCHEMBL10271336 0.67 KDM4E (0.55) SMN1; SMN2CYP1A2CYP2C9ADORA1
SCHEMBL27017989 0.67 KMO (0.41) FLT3
SCHEMBL22010374 0.67 KMO (0.44) SMN1; SMN2
SCHEMBL30892721 0.66 ADORA2A (0.39) SMN1; SMN2CYP1A2CYP2C9ADORA1
SCHEMBL13779843 0.65
SCHEMBL503382 0.65
SCHEMBL4709224 0.65 GSK3B (0.50) SMN1; SMN2PDE3BPDE3ACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2033963-B1 Substituted 2-(diaza-bicyclo-alkyl)-pyrimidone derivatives SANOFI AVENTIS (FR) 2011-02-16 EP claimed
EP-2033963-A1 Substituted 2-(diaza-bicyclo-alkyl)-pyrimidone derivatives Sanofi-Aventis (FR) 2009-03-11 EP claimed