SCHEMBL11308142

SCHEMBL11308142

CCOC(=O)Nc1c(C)cc(C(=O)CBr)cc1Br

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 8/20 0.46
SMN1; SMN2 Q16637 1/20 0.42
KDM4E B2RXH2 2/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
F2R P25116 1/20 0.40
GLA P06280 1/20 0.39
POLB P06746 1/20 0.39
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
GSK3B P49841 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11035760 0.86 NLRP3 (0.48) NLRP3SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL11326131 0.83 NLRP3 (0.41) NLRP3SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL11546525 0.80 NLRP3 (0.49) NLRP3SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL11545247 0.79 GSK3B (0.42) SMN1; SMN2KDM4EHPGDPOLBHSD17B10
SCHEMBL1000325 0.76 NLRP3 (0.59) NLRP3SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL11547384 0.73 GSK3B (0.37) NLRP3KDM4EKMT2AMEN1HPGD
SCHEMBL11552739 0.72 GSK3B (0.44) HPGDLMNAGSK3B
SCHEMBL26588963 0.72 NLRP3 (0.78) NLRP3SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL30741281 0.71 NLRP3 (0.48) NLRP3SMN1; SMN2KDM4ECYP1A2CYP2C9
SCHEMBL11956604 0.71 GSK3B (0.54) KMT2AMEN1MAPTGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0057900-A1 Animal feed additive for improving growth Dr. Karl Thomae GmbH (DE) 1982-08-18 EP disclosed
EP-0008715-B1 PHENYLETHANOLAMINES FOR USE IN COMBATTING INFLAMMATORY CONDITIONS Dr. Karl Thomae GmbH (DE) 1981-11-25 EP disclosed
US-4244967-A ANTIIFLAMMATORY AND ANTIRHEUMATIC PROPERTIES BOEHRINGER INGELHEIM GMBH (DE) 1981-01-13 US disclosed
US-4214001-A ANALGESICS, ANTISPASMODICS AND ANTIASTHMATICS BOEHRINGER INGELHEIM GMBH (DE) 1980-07-22 US disclosed
EP-0008715-A1 Phenylethanolamines for use in combatting inflammatory conditions Dr. Karl Thomae GmbH (DE) 1980-03-19 EP disclosed