SCHEMBL11316248

SCHEMBL11316248

N=C(N)NC(=O)Nc1c(Cl)cccc1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.43
POLB P06746 1/20 0.40
MAPT P10636 1/20 0.40
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
HTR2B P41595 1/20 0.38
CXCR1 P25024 1/20 0.37
CXCR2 P25025 1/20 0.37
PKM P14618 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TYK2 P29597 1/20 0.36
KDM4E B2RXH2 2/20 0.35
LMNA P02545 2/20 0.35
CACNA1C Q13936 1/20 0.35
SCN5A Q14524 1/20 0.35
ALDH1A1 P00352 1/20 0.35
F2 P00734 1/20 0.35
F10 P00742 1/20 0.35
PLAU P00749 1/20 0.35
PLAT P00750 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11139508 0.89 DRD2 (0.42) CYP1A2POLBDRD2HTR2AHTR2B
SCHEMBL11057728 0.89 CYP1A2 (0.49) CYP1A2POLBDRD2HTR2AHTR2B
Hydrochloric Acid SCHEMBL11320569 0.87 CYP1A2 (0.47) CYP1A2POLBDRD2HTR2AHTR2B
SCHEMBL11883002 0.84 GAA (0.37) CXCR1CXCR2TYK2LMNAF2
SCHEMBL11054621 0.82 POLB (0.41) CYP1A2POLBMAPTNPSR1TYK2
SCHEMBL11307694 0.82 KMT2A (0.44) MAPTDRD2HTR2AHTR2BPKM
SCHEMBL11093150 0.82 CYP1A2 (0.43) CYP1A2CXCR1CXCR2TYK2LMNA
SCHEMBL11056409 0.82 KMT2A (0.47) CYP1A2DRD2HTR2AHTR2BNPSR1
SCHEMBL7168279 0.82 DRD2 (0.55) CYP1A2POLBMAPTDRD2HTR2A
SCHEMBL7168272 0.82 DRD2 (0.55) CYP1A2POLBDRD2HTR2AHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4283555-A Amidinoureas WILLIAM H. RORER, INC. (US) 1981-08-11 US claimed
US-4219567-A ANTIULCER AGENTS WILLIAM H. RORER, INC. (US) 1980-08-26 US claimed
US-4183956-A Method for treating gastrointestinal spasms, gastrointestinal hyperacidity and hypertensive disorders with amidinoureas WILLIAM H. RORER, INC. (US) 1980-01-15 US claimed
US-4283555-A Amidinoureas WILLIAM H. RORER, INC. (US) 1981-08-11 US disclosed
US-4219567-A ANTIULCER AGENTS WILLIAM H. RORER, INC. (US) 1980-08-26 US disclosed
US-4183956-A Method for treating gastrointestinal spasms, gastrointestinal hyperacidity and hypertensive disorders with amidinoureas WILLIAM H. RORER, INC. (US) 1980-01-15 US disclosed