SCHEMBL11320142

SCHEMBL11320142

COCCc1ccc(OCC(CNC(C)C)OC(=O)/C=C/C(=O)OC(CNC(C)C)COc2ccc(CCOC)cc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 3/20 0.63
ADRB2 P07550 2/20 0.63
CYP2D6 P10635 2/20 0.63
NR3C1 P04150 1/20 0.63
ADRA1A P35348 1/20 0.63
CYP2J2 P51589 1/20 0.63
PDE4D Q08499 1/20 0.63
NPY1R P25929 1/20 0.61
NPY2R P49146 1/20 0.61
PMP22 Q01453 1/20 0.61
NPSR1 Q6W5P4 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
ABCB1 P08183 1/20 0.46
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9636570 0.92 ADRB1 (0.56) ADRB1ADRB2CYP2D6NR3C1ADRA1A
SCHEMBL7274537 0.92 ADRB1 (0.56) ADRB1ADRB2CYP2D6NR3C1ADRA1A
SCHEMBL8892157 0.88 ADRB1 (0.66) ADRB1ADRB2CYP2D6NR3C1ADRA1A
SCHEMBL2473791 0.87 ADRB1 (0.65) ADRB1ADRB2CYP2D6NR3C1ADRA1A
SCHEMBL4456681 0.86 NPY1R (0.67) ADRB1ADRB2CYP2D6NR3C1ADRA1A
Fumaric Acid SCHEMBL10909713 0.85 NPY1R (0.58) ADRB1ADRB2CYP2D6NR3C1ADRA1A
SCHEMBL20887451 0.84 ADRB1 (0.61) ADRB1ADRB2CYP2D6NR3C1ADRA1A
SCHEMBL7286484 0.83 NPY1R (0.75) ADRB1ADRB2CYP2D6NR3C1ADRA1A
SCHEMBL11307344 0.82 ADRB2 (0.43) ADRB1ADRB2CYP2D6ADRA1APMP22
SCHEMBL9799095 0.82 NPY1R (0.59) ADRB1ADRB2CYP2D6NR3C1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4303637-A Medication indicated for ocular hypertension ALZA CORPORATION (US) 1981-12-01 US disclosed
EP-0037622-A2 Drug delivery insert for controlled ocular therapy ALZA CORPORATION (US) 1981-10-14 EP disclosed