SCHEMBL11322262

SCHEMBL11322262

COc1ccc(NC=O)c(CCc2ccccn2)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.48
RAB9A P51151 3/20 0.47
NPC1 O15118 2/20 0.47
MTNR1A P48039 1/20 0.46
MTNR1B P49286 1/20 0.46
ABCB1 P08183 1/20 0.44
HTR1A P08908 1/20 0.44
DRD2 P14416 1/20 0.44
MEN1 O00255 2/20 0.43
MAPT P10636 2/20 0.42
GAA P10253 2/20 0.42
ACP1 P24666 1/20 0.42
SYK P43405 2/20 0.42
TSHR P16473 1/20 0.41
GRM5 P41594 1/20 0.41
TP53 P04637 1/20 0.41
ALDH1A1 P00352 2/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11329237 0.80 HRH3 (0.44) ABCB1HTR1ADRD2ALDH1A1LMNA
SCHEMBL11319599 0.77 NPC1 (0.50) KMT2ARAB9ANPC1MTNR1AMTNR1B
SCHEMBL9947244 0.75 OR51E2 (0.50) KMT2ADRD2TSHRALDH1A1LMNA
Iodide SCHEMBL11324465 0.74 OR51E2 (0.38) KMT2ARAB9ANPC1MTNR1AMTNR1B
SCHEMBL5216491 0.73 OR51E2 (0.51) DRD2MAPTTSHRALDH1A1OR51E2
SCHEMBL13955392 0.72 TSHR (0.47) KMT2ARAB9ANPC1MTNR1AMTNR1B
SCHEMBL18971459 0.71 MTNR1A (0.52) KMT2ARAB9ANPC1MTNR1AMTNR1B
SCHEMBL10752732 0.71 NPC1 (0.64) KMT2ARAB9ANPC1HTR1AMAPT
SCHEMBL29167655 0.70 SYK (0.52) KMT2ARAB9ANPC1MTNR1AMTNR1B
SCHEMBL13936668 0.70 TSHR (0.45) KMT2ARAB9ANPC1MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE30812-E ANTIARRHTHMIA AGENTS MEAD JOHNSON & COMPANY (US) 1981-12-01 US disclosed
US-RE30811-E SEROTONIN ANTAGONISTS, ANTIARRHYTHMIA AGENTS MEAD JOHNSON & COMPANY (US) 1981-12-01 US disclosed
US-4064254-A ANTIARRHYTHMIC AND ANTISEROTONINE AGENTS MEAD JOHNSON & COMPANY (US) 1977-12-20 US disclosed
US-4000143-A ANTIARRHYTHMIC AND ANTISEROTONIN AGENTS MEAD JOHNSON & COMPANY (US) 1976-12-28 US disclosed
US-3931195-A ANTIARRHYTHMIA, ANTISEROTONIN MEAD JOHNSON & COMPANY (US) 1976-01-06 US disclosed