SCHEMBL11340409

SCHEMBL11340409

Cc1c(C#N)c(N)n(-c2ccc(F)cc2)c1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.49
ALDH1A1 P00352 7/20 0.43
HPGD P15428 4/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
GAA P10253 2/20 0.43
MAPT P10636 2/20 0.43
RXFP1 Q9HBX9 2/20 0.41
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
TSHR P16473 2/20 0.39
PTGS2 P35354 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
MITF O75030 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
TP53 P04637 1/20 0.37
PIK3CD O00329 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11345308 0.87 ALDH1A1 (0.56) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL11339280 0.84 KDM4E (0.54) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL11340384 0.83 ALDH1A1 (0.57) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL11345226 0.81 ALDH1A1 (0.48) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL11332732 0.78 ALDH1A1 (0.51) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL11335662 0.77 L3MBTL1 (0.44) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL11494325 0.73 HTT (0.38) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL3259352 0.73 KDM4E (0.56) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL11339426 0.71 ALDH1A1 (0.44) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL11362989 0.70 ALDH1A1 (0.44) KDM4EALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0005205-B1 SUBSTITUTED 5.6-DIMETHYLPYRROLO(2,3-D)PYRIMIDINES, METHODS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM Troponwerke GmbH & Co. KG (DE) 1981-09-09 EP disclosed
US-4229453-A ANTIINFLAMMATORY AGENTS, SEDATIVES, ANTICONVULSANTS BAYER AKTIENGESELLSCHAFT (DE) 1980-10-21 US disclosed