SCHEMBL1134529

SCHEMBL1134529

Brc1cncc(Br)c1.Brc1cncc(NCc2ccccc2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.52
LTA4H P09960 1/20 0.47
KCNH2 Q12809 1/20 0.46
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
HTT P42858 2/20 0.43
KDR P35968 1/20 0.43
PTPN1 P18031 1/20 0.43
PTPN11 Q06124 1/20 0.43
PDGFRB P09619 1/20 0.43
PDGFRA P16234 1/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
GABRA5 P31644 1/20 0.43
GABRA3 P34903 1/20 0.43
DHFR P00374 1/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2064845 0.98 SMN1; SMN2 (0.54) SMN1; SMN2LTA4HKCNH2CHRNB2CHRNA4
SCHEMBL22191644 0.89 FFAR1 (0.47) SMN1; SMN2KCNH2GABRG2GABRB3GABRA5
SCHEMBL22191444 0.85 GAA (0.47) SMN1; SMN2HTTKDRALDH1A1KMT2A
SCHEMBL22191758 0.84 LTA4H (0.61) LTA4HHTTMEN1ALDH1A1KMT2A
SCHEMBL5386751 0.82 HTT (0.52) SMN1; SMN2HTTPTPN1PTPN11ALDH1A1
SCHEMBL22191439 0.82 KDM4E (0.46) KCNH2ALDH1A1HPGDLMNA
SCHEMBL4651084 0.82 HTR7 (0.58) SMN1; SMN2KCNH2KDRPOLB
SCHEMBL4147020 0.82 KDM4E (0.46) SMN1; SMN2KDRMEN1ALDH1A1KMT2A
SCHEMBL1713545 0.81 INSR (0.48) SMN1; SMN2GABRG2GABRB3GABRA5GABRA3
SCHEMBL6122773 0.81 CCNT1 (0.49) KCNH2MEN1ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2285810-A1 SELECTIVE LIGANDS FOR THE NEURONAL NICOTINIC RECEPTORS AND USES THEREOF Abbott Laboratories (US) 2011-02-23 EP disclosed
WO-2009137308-A1 SELECTIVE LIGANDS FOR THE NEURONAL NICOTINIC RECEPTORS AND USES THEREOF ABBOTT LABORATORIES (US) 2009-11-12 WO disclosed