SCHEMBL11348484

SCHEMBL11348484

O=C(C[N+](=O)[O-])Nc1ccc(Br)c(Cl)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 7/20 0.61
KMT2A Q03164 7/20 0.61
LMNA P02545 5/20 0.61
ALDH1A1 P00352 5/20 0.61
HPGD P15428 5/20 0.61
GAA P10253 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
MAPT P10636 6/20 0.55
SMN1; SMN2 Q16637 3/20 0.52
HTT P42858 2/20 0.52
NPC1 O15118 2/20 0.52
ALOX15 P16050 2/20 0.51
ALOX12 P18054 2/20 0.51
F13A1 P00488 1/20 0.49
TGM2 P21980 1/20 0.49
RAB9A P51151 2/20 0.47
PKM P14618 1/20 0.47
TP53 P04637 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP3A4 P08684 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11347529 0.86 KMT2A (0.43) MEN1KMT2ALMNAALDH1A1HPGD
SCHEMBL8512871 0.86 CYP3A4 (0.61) MEN1KMT2ALMNAALDH1A1L3MBTL1
SCHEMBL10995578 0.82 TSHR (0.64) MEN1KMT2ALMNAALDH1A1HPGD
SCHEMBL27546640 0.82 HPGD (0.61) MEN1KMT2ALMNAALDH1A1HPGD
SCHEMBL20165835 0.80 CYP3A4 (0.57) MEN1KMT2ALMNAALDH1A1GAA
SCHEMBL8125102 0.80 MEN1 (0.69) MEN1KMT2ALMNAALDH1A1HPGD
SCHEMBL5491596 0.79 ALDH1A1 (0.60) MEN1KMT2ALMNAALDH1A1HPGD
SCHEMBL2933871 0.78 KMT2A (0.63) MEN1KMT2ALMNAALDH1A1HPGD
SCHEMBL11763476 0.78 KMT2A (0.59) MEN1KMT2ALMNAALDH1A1HPGD
SCHEMBL14779722 0.77 MEN1 (0.80) MEN1KMT2ALMNAALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0029658-A1 Salts of dihalo-2-quinoxaline carboxylic acids, their preparation and pharmaceutical formulations containing them ELI LILLY AND COMPANY (US) 1981-06-03 EP disclosed
US-4264600-A VIRICIDES ELI LILLY AND COMPANY (US) 1981-04-28 US disclosed
US-4252954-A VIRICIDES ELI LILLY AND COMPANY (US) 1981-02-24 US disclosed
EP-0010426-A1 Pharmaceutical composition containing 3,4-dihydro-3-oxo-2-quinoxalines, novel such quinoxalines and processes for the production thereof ELI LILLY AND COMPANY (US) 1980-04-30 EP disclosed