SCHEMBL11348807

SCHEMBL11348807

COc1cccc(C(=O)CC2CCCN2)c1

nearest known ligand 0.59

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.50
CHRM2 P08172 1/20 0.48
CHRM1 P11229 1/20 0.48
CHRM3 P20309 1/20 0.48
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
KHK P50053 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
CDYL2 Q8N8U2 1/20 0.47
CDYL Q9Y232 1/20 0.47
CHRNB4 P30926 1/20 0.46
CHRNA3 P32297 1/20 0.46
PARP1 P09874 1/20 0.46
CTNNB1 P35222 2/20 0.45
WNT3A P56704 2/20 0.45
HSD11B1 P28845 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL11382277 0.99 GHSR (0.49) GHSRCHRM2CHRM1CHRM3CES2
SCHEMBL465887 0.84 RELA (0.47) GHSRKHK
SCHEMBL11343167 0.79 KHK (0.52) GHSRCES1KHKMEN1KMT2A
Bromide SCHEMBL11099888 0.78 CHRM2 (0.49) CHRM2CHRM1CHRM3CES2CES1
SCHEMBL21848527 0.76 KHK (0.45) KHK
SCHEMBL11164963 0.76 CTNNB1 (0.47) CHRM2CHRM1CHRM3CES2CES1
SCHEMBL29039262 0.75 CHRNB4 (0.63) CHRNB4CHRNA3
SCHEMBL26999492 0.75 CHRNB4 (0.63) CHRNB4CHRNA3
SCHEMBL11807455 0.75 MEN1 (0.49) MEN1KMT2ACHRNB4CHRNA3HSD11B1
SCHEMBL7860033 0.75 POLB (0.54) KHKKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0002672-B1 SUBSTITUTED PYRROLIDINES, PROCESS FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1981-08-26 EP disclosed
US-4198424-A ANALGESICS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1980-04-15 US disclosed
EP-0002672-A2 Substituted pyrrolidines, process for their preparation and medicaments containing them Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1979-07-11 EP disclosed