SCHEMBL11349132

SCHEMBL11349132

Cc1ccc(-n2nnc(C(=O)O)c2N)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.56
CA2 P00918 3/20 0.56
CA4 P22748 3/20 0.56
CA9 Q16790 3/20 0.56
TP53 P04637 1/20 0.56
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
ALDH1A1 P00352 3/20 0.56
CYP1A2 P05177 2/20 0.56
CYP2C19 P33261 2/20 0.56
MAPT P10636 2/20 0.56
HTT P42858 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.52
MAPK1 P28482 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
GAA P10253 1/20 0.50
PTGS2 P35354 1/20 0.50
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
KDM4E B2RXH2 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4789300 0.85 TP53 (0.69) CA1CA2CA4CA9TP53
SCHEMBL20604184 0.83 HTT (0.78) CA1CA2CA4CA9TP53
SCHEMBL10986951 0.81 TP53 (0.68) CA2TP53ALDH1A1CYP1A2HTT
SCHEMBL11333929 0.81 SMN1; SMN2 (0.79) CA1CA2CA4CA9TP53
SCHEMBL30808868 0.78 HTT (0.53) CA1CA2CA4CA9TP53
SCHEMBL27848899 0.77 CA1 (0.61) CA1CA2CA4CA9ALDH1A1
SCHEMBL31755988 0.76 DCTPP1 (0.51) CA1CA2CA4CA9TP53
SCHEMBL10983505 0.76 SMN1; SMN2 (0.67) CA1CA2CA4CA9TP53
SCHEMBL19501329 0.75 CA2 (0.58) CA1CA2CA4CA9TP53
SCHEMBL12088095 0.75 TP53 (0.70) CA1CA2CA9TP53MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0002562-B1 TRIAZOLO-QUINOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR PHARMACEUTICAL USE BEECHAM GROUP PLC (GB) 1981-05-20 EP disclosed
EP-0002562-A1 Triazolo-quinoline derivatives, processes for their preparation and their pharmaceutical use BEECHAM GROUP PLC (GB) 1979-06-27 EP disclosed