SCHEMBL11360366

SCHEMBL11360366

NNc1cc2c(nn1)CC1CCC2N1C(=O)c1ccccc1Cl

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.37
PTGS1 P23219 1/20 0.36
GAA P10253 1/20 0.36
RAB9A P51151 1/20 0.36
GPR65 Q8IYL9 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
FFAR2 O15552 1/20 0.34
PAK1 Q13153 1/20 0.34
P2RX7 Q99572 2/20 0.34
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CCNA1 P78396 1/20 0.33
EPHX2 P34913 1/20 0.33
F2 P00734 1/20 0.33
MGLL Q99685 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11363313 0.73 ALDH1A1 (0.44) PTGS1EPHX2ALDH1A1
SCHEMBL11085199 0.68 PTGS1 (0.72) KMT2APTGS1RAB9AP2RX7ALDH1A1
SCHEMBL19014041 0.62 KMT2A (0.50) KMT2AGAARAB9ATDP1P2RX7
SCHEMBL19014514 0.59 P2RX7 (0.49) GAARAB9ATDP1P2RX7MGLL
SCHEMBL20682253 0.59 KDM4E (0.46) KMT2AGAARAB9ATDP1P2RX7
SCHEMBL11117707 0.58 PTGS1 (0.70) KMT2APTGS1GAARAB9AP2RX7
SCHEMBL11360399 0.58 JAK3 (0.32) GPR65MGLL
SCHEMBL11351452 0.58 KMT2A (0.33) KMT2AGPR65MGLL
SCHEMBL10243903 0.57 HSD11B1 (0.51) KMT2AGAARAB9AP2RX7MGLL
SCHEMBL17350802 0.57 HSD11B1 (0.51) KMT2AGAARAB9AP2RX7MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4277472-A 3,6-Disubstituted-5,7-(lower alkano)-5,6,7,8-tetrahydropyrido(4,3-C)pyridazines; their intermediates, preparation, antihypertensive use and compositions BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1981-07-07 US disclosed