SCHEMBL11360802

SCHEMBL11360802

O=C1NC(c2ccccc2)C2(CCN(C(=O)OCc3ccccc3)CC2)O1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
KDM1A O60341 2/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
CYP2C19 P33261 1/20 0.47
ENPP2 Q13822 2/20 0.46
ATXN2 Q99700 2/20 0.46
OPRK1 P41145 4/20 0.45
GRIN2B Q13224 1/20 0.43
HTT P42858 1/20 0.43
HTR1A P08908 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
HTR2C P28335 1/20 0.43
SLC6A3 Q01959 1/20 0.43
CCR5 P51681 2/20 0.43
HDAC3 O15379 1/20 0.43
HDAC1 Q13547 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11369993 0.85 MEN1 (0.50) MEN1KMT2ANPSR1KDM1ASMN1; SMN2
SCHEMBL4458368 0.81 CCR5 (0.49) MEN1KMT2ANPSR1KDM1ASMN1; SMN2
SCHEMBL1488930 0.76 HTR2C (0.48) MEN1KMT2ANPSR1SMN1; SMN2NPC1
SCHEMBL4134071 0.76 MEN1 (0.55) MEN1KMT2ANPSR1KDM1ASMN1; SMN2
SCHEMBL11368285 0.76 LMNA (0.57) MEN1KMT2ANPSR1KDM1ASMN1; SMN2
SCHEMBL11361449 0.73 MEN1 (0.52) MEN1KMT2ANPSR1KDM1ASMN1; SMN2
SCHEMBL23859760 0.73 SMN1; SMN2 (0.56) MEN1KMT2ANPSR1KDM1ASMN1; SMN2
SCHEMBL18075928 0.73 SMN1; SMN2 (0.51) MEN1KMT2ANPSR1KDM1ASMN1; SMN2
SCHEMBL934263 0.73 MEN1 (0.64) MEN1KMT2ANPSR1KDM1ASMN1; SMN2
SCHEMBL2425665 0.73 MEN1 (0.54) MEN1KMT2ANPSR1KDM1ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4255432-A ANTIHYPERTENSIVE AGENTS, ANTIHISTAMINES, BRONCHODILATOR AGENTS, ANTIVASOSPASTIC AGENTS SYNTEX (U.S.A.) INC. (US) 1981-03-10 US disclosed
US-4244961-A 1-Oxa-3,8-diazaspiro[4.5]decan-2-ones antihypertensive agents SYNTEX (U.S.A.) INC. (US) 1981-01-13 US disclosed