SCHEMBL1138720

SCHEMBL1138720

COC(=O)c1ccc(NC(=O)c2cc(Cl)ccc2NS(=O)(=O)c2ccccc2)cc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.76
MEN1 O00255 3/20 0.76
KMT2A Q03164 3/20 0.76
LMNA P02545 2/20 0.76
ALDH1A1 P00352 2/20 0.76
KDM4E B2RXH2 1/20 0.76
CYP3A4 P08684 1/20 0.76
CYP2D6 P10635 1/20 0.76
CYP2C9 P11712 1/20 0.76
HPGD P15428 1/20 0.76
CRHBP P24387 1/20 0.76
CYP2C19 P33261 1/20 0.76
CRHR2 Q13324 1/20 0.76
SMN1; SMN2 Q16637 1/20 0.76
NOD2 Q9HC29 1/20 0.76
GPR27 Q9NS67 7/20 0.59
AVPR2 P30518 2/20 0.59
SLC10A6 Q3KNW5 2/20 0.58
SLC10A2 Q12908 1/20 0.58
SLC10A1 Q14973 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1138705 0.89 SLC10A6 (0.63) HTTMEN1KMT2ALMNAALDH1A1
SCHEMBL7109904 0.85 MEN1 (0.55) HTTMEN1KMT2ALMNAALDH1A1
SCHEMBL5124913 0.84 SLC10A6 (0.57) HTTMEN1KMT2ALMNAALDH1A1
SCHEMBL1138698 0.84 KDM4E (0.64) HTTMEN1KMT2ALMNAKDM4E
SCHEMBL10249599 0.84 GPR27 (0.66) GPR27AVPR2SLC10A6SLC10A2SLC10A1
SCHEMBL1139427 0.84 KMT2A (0.57) HTTMEN1KMT2ALMNAALDH1A1
SCHEMBL5120009 0.83 SLC10A6 (0.62) HTTMEN1KMT2ALMNAALDH1A1
SCHEMBL6860504 0.83 SLC10A6 (0.59) HTTMEN1KMT2ALMNAALDH1A1
SCHEMBL6862400 0.83 SLC10A6 (0.71) MEN1KMT2AKDM4EGPR27AVPR2
SCHEMBL6754585 0.83 SLC10A6 (0.81) MEN1KMT2ALMNAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0947500-B1 SULFONAMIDE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2011-02-23 EP disclosed
EP-0947500-B1 SULFONAMIDE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2011-02-23 EP disclosed
CN-1213019-C Sulfonamide and carboxamide derivatives and drugs containing same as active ingredient ONO PHARMACEUTICAL CO (JP) 2005-08-03 CN disclosed
US-6790866-B2 SUCH AS 4-(2-PHENYLSULFONYLAMINO-5-CHLOROBENZOYLAMINO)BENZOIC ACID FOR USE AS PROSTAGLANDIN E2 ANTAGONIST OR AGONIST; FOR INHIBITION OF UTERINE CONTRACTION, ANALGESICS, ANTIDIARRHEALS, SLEEP INDUCERS, AND/OR FOR INCREASE OF VESICAL CAPACITY ONO PHARMACEUTICAL CO., LTD. (JP) 2004-09-14 US disclosed
US-20030060460-A1 Such as 4-(2-phenylsulfonylamino-5-chlorobenzoylamino)benzoic acid for use as prostaglandin E2 antagonist or agonist; for inhibition of uterine contraction, analgesics, antidiarrheals, sleep inducers, and/or for increase of vesical capacity OHUCHIDA SHUICHI (JP) 2003-03-27 US disclosed
US-6448290-B1 PROSTAGLANDIN E2 ANTAGONIST OR AGONIST; INHIBITION OF UTERINE CONTRACTION, ANALGESICS, ANTIDIARRHEALS, SLEEP INDUCERS, INCREASING VESICAL CAPACITY, CATHARTIC, SUPPRESSION OF GASTRIC ACID SECRETION, ANTIHYPERTENSIVE, DIURETIC AGENTS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-09-10 US disclosed
EP-0947500-A1 SULFONAMIDE AND CARBOXAMIDE DERIVATIVES AND DRUGS CONTAINING THE SAME AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO., LTD. (JP) 1999-10-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030060460-A1 Such as 4-(2-phenylsulfonylamino-5-chlorobenzoylamino)benzoic acid for use as prostaglandin E2 antagonist or agonist; for inhibition of uterine contraction, analgesics, antidiarrheals, sleep inducers, and/or for increase of vesical capacity CNR1, HCAR1, HCAR2 HTT 3078/4885MEN1 4832/4885KMT2A 1316/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.