SCHEMBL11429463

SCHEMBL11429463

CCC(=O)N[C@@H](C)C(=O)N1CCC[C@H]1C(=O)NC1CCCCCCC1

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
POLB P06746 2/20 0.49
NPSR1 Q6W5P4 1/20 0.48
TSHR P16473 2/20 0.45
MAPK1 P28482 1/20 0.43
ALDH1A1 P00352 2/20 0.43
GAA P10253 2/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
EPHX2 P34913 2/20 0.41
REN P00797 2/20 0.41
ACE P12821 1/20 0.41
EPHX1 P07099 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11431101 1.00 KDM4E (0.54) KDM4ESMN1; SMN2POLBNPSR1TSHR
SCHEMBL11430017 1.00 KDM4E (0.54) KDM4ESMN1; SMN2POLBNPSR1TSHR
SCHEMBL11429475 0.99 KDM4E (0.52) KDM4ESMN1; SMN2POLBNPSR1TSHR
SCHEMBL11516951 0.86 ACE (0.46) KDM4ERENACE
SCHEMBL11517034 0.85 ACE (0.45) KDM4ERENACE
SCHEMBL18681285 0.84 ACE (0.44) KDM4ERENACE
SCHEMBL11519144 0.84 FKBP5 (0.44) KDM4EPOLBRENACE
SCHEMBL11431773 0.82 ACE (0.61) KDM4ERENACE
SCHEMBL11429550 0.79 NPSR1 (0.52) POLBNPSR1TSHRRENACE
Bromide SCHEMBL11441971 0.78 KDM4E (0.61) KDM4ESMN1; SMN2POLBNPSR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4187216-A ELASTASE INHIBITORS HOFFMANN-LA ROCHE INC. (US) 1980-02-05 US claimed
US-4187216-A ELASTASE INHIBITORS HOFFMANN-LA ROCHE INC. (US) 1980-02-05 US disclosed