SCHEMBL11517034

SCHEMBL11517034

CCC(=O)N[C@@H](C)C(=O)N1CCC[C@H]1C(=O)NC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACE P12821 7/20 0.45
REN P00797 4/20 0.45
PREP P48147 1/20 0.43
FAP Q12884 1/20 0.43
MMP1 P03956 3/20 0.42
MMP13 P45452 3/20 0.42
ADAM17 P78536 3/20 0.42
MMP3 P08254 2/20 0.42
KDM4E B2RXH2 1/20 0.42
F2 P00734 1/20 0.42
LMNA P02545 1/20 0.42
LTA4H P09960 1/20 0.42
MAPT P10636 1/20 0.42
PEPD P12955 1/20 0.42
ALOX15 P16050 1/20 0.42
PTGS1 P23219 1/20 0.42
HTR2A P28223 1/20 0.42
PTGS2 P35354 1/20 0.42
HRH1 P35367 1/20 0.42
THPO P40225 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11516951 0.90 ACE (0.46) ACERENPREPFAPKDM4E
SCHEMBL18681285 0.88 ACE (0.44) ACERENPREPFAPKDM4E
SCHEMBL11519144 0.88 FKBP5 (0.44) ACERENPREPFAPKDM4E
SCHEMBL11431773 0.86 ACE (0.61) ACERENKDM4EF2LMNA
SCHEMBL11429475 0.86 KDM4E (0.52) ACERENPREPFAPKDM4E
SCHEMBL11429463 0.85 KDM4E (0.54) ACERENKDM4E
SCHEMBL11430017 0.85 KDM4E (0.54) ACERENKDM4E
SCHEMBL11431101 0.85 KDM4E (0.54) ACERENKDM4E
SCHEMBL11429550 0.83 NPSR1 (0.52) ACEREN
SCHEMBL10658127 0.82 ACE (0.56) ACERENKDM4EF2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4176116-A ELASTASE ENZYME INHIBITORS HOFFMANN-LA ROCHE INC. (US) 1979-11-27 US claimed
US-4176116-A ELASTASE ENZYME INHIBITORS HOFFMANN-LA ROCHE INC. (US) 1979-11-27 US disclosed