SCHEMBL114463

SCHEMBL114463

NC(=O)OCc1ccccc1Br

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 1/20 0.57
IDO1 P14902 2/20 0.57
MMP1 P03956 1/20 0.53
MMP2 P08253 1/20 0.53
MMP9 P14780 1/20 0.53
MMP12 P39900 1/20 0.53
ALDH1A1 P00352 5/20 0.50
MAPT P10636 3/20 0.50
RAB9A P51151 2/20 0.50
KMT2A Q03164 2/20 0.50
PKM P14618 2/20 0.50
POLB P06746 1/20 0.50
NPC1 O15118 1/20 0.47
FFAR4 Q5NUL3 2/20 0.45
FFAR1 O14842 1/20 0.45
TAAR1 Q96RJ0 1/20 0.44
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29501710 0.86 SMN1; SMN2 (0.48) PARP10IDO1ALDH1A1PKMCYP1A2
SCHEMBL7765576 0.84 MAPT (0.56) PARP10IDO1MMP1MMP2MMP9
SCHEMBL7760184 0.82 ALDH1A1 (0.56) PARP10IDO1MMP1MMP2MMP9
SCHEMBL6702870 0.82 MMP1 (0.54) PARP10IDO1MMP1MMP2MMP9
SCHEMBL30429390 0.82 ALDH1A1 (0.56) PARP10IDO1MMP1MMP2MMP9
SCHEMBL29272771 0.82 MMP1 (0.41) PARP10IDO1MMP1MMP2MMP9
SCHEMBL2548713 0.81 TAAR1 (0.50) PARP10IDO1MMP1MMP2MMP9
SCHEMBL10800307 0.81 ALDH1A1 (0.56) PARP10IDO1MMP1MMP2MMP9
SCHEMBL777869 0.81 MAPT (0.57) PARP10IDO1MMP1MMP2MMP9
SCHEMBL6176778 0.81 ALDH1A1 (0.55) PARP10IDO1MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 508 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250257031-A1 PROCESS FOR THE PRODUCTION OF SUBSTITUTED 2-[2-(PHENYL)ETHYLAMINO]ALKANEAMIDE DERIVATIVES NEWRON PHARMACEUTICALS S.P.A. (IT) 2025-08-14 US claimed
US-12291495-B2 Process for the production of substituted 2-[2-(phenyl)ethylamino] alkaneamide derivatives NEWRON PHARMACEUTICALS S.P.A. (IT) 2025-05-06 US claimed
US-20220185766-A1 PROCESS FOR THE PRODUCTION OF SUBSTITUTED 2-[2-(PHENYL)ETHYLAMINO]ALKANEAMIDE DERIVATIVES NEWRON PHARMACEUTICALS S.P.A. (IT) 2022-06-16 US claimed
EP-3956296-A1 PROCESS FOR THE PRODUCTION OF SUBSTITUTED 2-[2-(PHENYL) ETHYLAMINO]ALKANEAMIDE DERIVATIVES Newron Pharmaceuticals S.p.A. (IT) 2022-02-23 EP claimed
WO-2020212352-A1 PROCESS FOR THE PRODUCTION OF SUBSTITUTED 2-[2-(PHENYL) ETHYLAMINO]ALKANEAMIDE DERIVATIVES NEWRON PHARMACEUTICALS S.P.A. (IT) 2020-10-22 WO claimed
EP-3725769-A1 PROCESS FOR THE PRODUCTION OF SUBSTITUTED 2-[2-(PHENYL) ETHYLAMINO]ALKANEAMIDE DERIVATIVES Newron Pharmaceuticals S.p.A. (IT) 2020-10-21 EP claimed
WO-2026089784-A2 COMPOUNDS AND COMPOSITIONS FOR CONJUGATION TO BIOLIGANDS FOR IMAGING AND RADIOPHARMACEUTICAL APPLICATIONS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2026-04-30 WO disclosed
US-20250257031-A1 PROCESS FOR THE PRODUCTION OF SUBSTITUTED 2-[2-(PHENYL)ETHYLAMINO]ALKANEAMIDE DERIVATIVES NEWRON PHARMACEUTICALS S.P.A. (IT) 2025-08-14 US disclosed
WO-2025151874-A1 INDOLE ALKALOID ANTIPLASMODIAL AGENTS AND PREPARATION THEREOF UNIVERSITY OF CENTRAL FLORIDA RESEARCH FOUNDATION, INC. (US) 2025-07-17 WO disclosed
US-12291495-B2 Process for the production of substituted 2-[2-(phenyl)ethylamino] alkaneamide derivatives NEWRON PHARMACEUTICALS S.P.A. (IT) 2025-05-06 US disclosed
WO-2025038960-A1 OLIGONUCLEOTIDES CONTAINING A LIGAND AT AN INTERNAL POSITION ADARX PHARMACEUTICALS, INC. (US) 2025-02-20 WO disclosed
US-12083186-B2 Methods for assembling scavenging particles NANOTICS, LLC (US) 2024-09-10 US disclosed
US-20240269319-A1 METHODS FOR ASSEMBLING SCAVENGING PARTICLES NANOTICS, LLC 2024-08-15 US disclosed
WO-2007117639-A9 SYNTHESIS OF TETRACYCLINES AND ANALOGUES THEREOF HARVARD COLLEGE (US) 2008-04-17 WO disclosed
WO-2007117639-A2 SYNTHESIS OF TETRACYCLINES AND ANALOGUES THEREOF THE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2007-10-18 WO disclosed
CN-101010336-A Peptide antibiotics and process for preparing same BIOSOURCE PHARM INC (US) 2007-08-01 CN disclosed
WO-2007013965-A2 SYNTHESIS OF SCABRONINES AND ANALOGUES THEREOF SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2007-02-01 WO disclosed
WO-2006138380-A2 AMINE-CONTAINING LIPIDS AND USES THEREOF MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2006-12-28 WO disclosed
WO-2006124902-A2 SYNTHESIS OF SALINOSPORAMIDE A AND ANALOGUES THEREOF SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2006-11-23 WO disclosed
WO-2006113615-A2 ANTI-MICROBIAL AGENTS AND USES THEREOF SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2006-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220185766-A1 PROCESS FOR THE PRODUCTION OF SUBSTITUTED 2-[2-(PHENYL)ETHYLAMINO]ALKANEAMIDE DERIVATIVES HRH3, CYP2A7, HRH4 PARP10 1129/4885IDO1 3435/4885MMP1 4111/4885
US-20250257031-A1 PROCESS FOR THE PRODUCTION OF SUBSTITUTED 2-[2-(PHENYL)ETHYLAMINO]ALKANEAMIDE DERIVATIVES HRH3, HRH4, H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16 PARP10 1275/4885IDO1 3371/4885MMP1 4095/4885
US-12291495-B2 Process for the production of substituted 2-[2-(phenyl)ethylamino] alkaneamide derivatives HRH3, CYP2A7, HRH4 PARP10 1129/4885IDO1 3435/4885MMP1 4111/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.