SCHEMBL11447474

SCHEMBL11447474

NC(=O)c1ccccc1NCCN1CCN(c2ccccc2N)CC1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.51
HTR7 P34969 3/20 0.51
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
DRD4 P21917 2/20 0.45
DRD2 P14416 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
NPC1 O15118 1/20 0.44
ADRA2C P18825 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methane SCHEMBL11602997 0.99 HTR1A (0.50) HTR1AHTR7HDAC3HDAC1DRD4
SCHEMBL11446752 0.93 HTR1A (0.54) HTR1AHTR7HDAC3HDAC1
SCHEMBL11605140 0.90 HTR1A (0.49) HTR1AHTR7HDAC3HDAC1DRD4
SCHEMBL11465718 0.88 HTR1A (0.51) HTR1AHTR7DRD4DRD2
SCHEMBL11447503 0.88 HTR1A (0.51) HTR1AHTR7DRD4DRD2CYP2D6
SCHEMBL11446726 0.87 HTR1A (0.53) HTR1AHTR7DRD4DRD2ALDH1A1
SCHEMBL11602992 0.85 HTR1A (0.49) HTR1AHTR7DRD4DRD2
SCHEMBL6933580 0.84 HTR1A (0.71) HTR1AHTR7DRD4DRD2
SCHEMBL11448262 0.84 HTR1A (0.58) HTR1AHTR7DRD2
SCHEMBL11447026 0.83 HTR7 (0.49) HTR1AHTR7KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4205173-A 1-Heterocyclic alkyl-1,2,3,4-tetrahydroquinazolinones and analgesic intermediates thereof PENNWALT CORPORATION (US) 1980-05-27 US disclosed
US-4085107-A ANALGESICS PENNWALT CORPORATION (US) 1978-04-18 US disclosed
US-4060526-A 1-Heterocyclic alkyl-1,2,3,4-tetrahydroquinazolinones and analgesic intermediates thereof PENNWALT CORPORATION (US) 1977-11-29 US disclosed