SCHEMBL11449484

SCHEMBL11449484

COc1cccc(OS(=O)(=O)c2ccc(Cl)c([N+](=O)[O-])c2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 3/20 0.56
ALPI P09923 3/20 0.56
VCAM1 P19320 11/20 0.53
NFE2L2 Q16236 1/20 0.50
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ALDH1A1 P00352 2/20 0.48
LMNA P02545 1/20 0.48
RAF1 P04049 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
MAPK1 P28482 1/20 0.48
GFER P55789 1/20 0.48
PAX8 Q06710 1/20 0.48
GPR17 Q13304 1/20 0.47
PIN1 Q13526 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11456478 0.88 ALPL (0.63) ALPLALPIVCAM1SMN1; SMN2ALDH1A1
SCHEMBL11448255 0.87 ALPL (0.59) ALPLALPIVCAM1CYP1A2CYP3A4
SCHEMBL11450417 0.87 CYP1A2 (0.61) ALPLALPIVCAM1CYP1A2CYP3A4
SCHEMBL11449495 0.86 ALPL (0.53) ALPLALPIVCAM1CYP1A2CYP3A4
SCHEMBL7179842 0.85 VCAM1 (0.62) ALPLALPIVCAM1
SCHEMBL11449191 0.85 ALDH1A1 (0.50) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL11450202 0.85 ALPL (0.54) ALPLALPIVCAM1CYP1A2CYP3A4
SCHEMBL11665975 0.84 APEX1 (0.60) ALPLALPINFE2L2CYP1A2CYP3A4
SCHEMBL11449208 0.82 ALPL (0.68) ALPLALPIVCAM1ALDH1A1
SCHEMBL11317864 0.81 ALPL (0.51) ALPLALPIVCAM1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4216161-A 3,4-Diaminophenyl sulfonic acid esters HOECHST AKTIENGESELLSCHAFT (DE) 1980-08-05 US disclosed
US-4069325-A 3-Carbalkoxyamino-1H-2,1,4-benzothiadiazine derivatives HOECHST AKTIENGESELLSCHAFT (DT) 1978-01-17 US disclosed
US-3996369-A Anthelmintically active 2-carbalkoxyamino benzimidazolyl-5(6)-sulfonic acid phenyl esters HOECHST AKTIENGESELLSCHAFT (DT) 1976-12-07 US disclosed