SCHEMBL11451997

SCHEMBL11451997

CCOC(=O)C1=C(C)NC(COC(C)=O)=C(C(=O)OCC)C1c1ccc(OC)cc1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.75
ALDH1A1 P00352 3/20 0.75
LMNA P02545 1/20 0.75
GAA P10253 1/20 0.75
HPGD P15428 1/20 0.75
HSD17B10 Q99714 1/20 0.75
TSHR P16473 1/20 0.60
SMN1; SMN2 Q16637 1/20 0.60
ABCC1 P33527 1/20 0.55
ADORA3 P0DMS8 2/20 0.53
CACNA1D Q01668 4/20 0.50
NPSR1 Q6W5P4 1/20 0.50
BCHE P06276 4/20 0.49
ACHE P22303 2/20 0.49
HRH3 Q9Y5N1 5/20 0.48
MEN1 O00255 1/20 0.48
MAPT P10636 1/20 0.48
MAPK1 P28482 1/20 0.48
KMT2A Q03164 1/20 0.48
CACNA1F O60840 3/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11452241 0.87 ABCC1 (0.74) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL11524111 0.87 KDM4E (0.81) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL11452070 0.87 ADORA3 (0.67) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL11470832 0.87 CACNA1D (0.59) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL7814802 0.86 KDM4E (1.00) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL11452254 0.80 DHFR (0.55) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL11461893 0.79 CACNA1B (0.53) KDM4EALDH1A1LMNATSHRSMN1; SMN2
SCHEMBL11459111 0.79 ABCC1 (0.55) KDM4EALDH1A1LMNATSHRSMN1; SMN2
SCHEMBL7817206 0.78 KDM4E (0.88) KDM4EALDH1A1LMNAGAAHPGD
SCHEMBL11735441 0.77 KDM4E (0.60) KDM4EALDH1A1LMNAGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4188395-A 1,4-Dihydropyridine derivatives substituted in the 2 position, and their use as medicaments BAYER AKTIENGESELLSCHAFT (DE) 1980-02-12 US disclosed