SCHEMBL114669

SCHEMBL114669

COc1ncc(-c2ccccc2N2CCN(C(C=O)n3ccc4c(Cl)ncnc43)CC2)cn1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.34
SLC2A1 P11166 11/20 0.33
SLC2A3 P11169 11/20 0.33
SLC2A2 P11168 9/20 0.33
TP53 P04637 2/20 0.33
LMNA P02545 2/20 0.32
DHFR P00374 1/20 0.32
HTR1A P08908 2/20 0.32
HTR7 P34969 2/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL111646 0.87 HTR1A (0.33) SLC2A1SLC2A3SLC2A2DHFRHTR1A
SCHEMBL113266 0.82 DHFR (0.35) MAPTSLC2A1SLC2A3SLC2A2LMNA
SCHEMBL115724 0.82 DHFR (0.33) MAPTDHFRHTR1AHTR7
SCHEMBL113317 0.81 DHFR (0.35) DHFRHTR1AHTR7
SCHEMBL116207 0.80 DHFR (0.33) LMNADHFRHTR1AHTR7
SCHEMBL114932 0.80 DHFR (0.35) SLC2A1SLC2A3SLC2A2DHFRHTR1A
SCHEMBL115607 0.78 HTR1A (0.37) MAPTLMNADHFRHTR1AHTR7
SCHEMBL116262 0.77 CXCR3 (0.35) DHFRHTR1AHTR7
SCHEMBL114668 0.77 CXCR3 (0.41) MAPTTP53LMNA
SCHEMBL113412 0.77 DHFR (0.35) DHFRHTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2424840-A1 CXCR3 RECEPTOR ANTAGONISTS Boehringer Ingelheim International GmbH (DE) 2012-03-07 EP disclosed
WO-2010126811-A1 CXCR3 RECEPTOR ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-11-04 WO disclosed