SCHEMBL11470978

SCHEMBL11470978

CC(C)N(CCC(C#N)(CCN(C)C)c1ccc(-c2ccccc2)cc1)C(C)C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.48
DRD3 P35462 3/20 0.48
CYP2D6 P10635 2/20 0.48
DRD2 P14416 2/20 0.48
DRD4 P21917 2/20 0.48
CYP3A4 P08684 2/20 0.40
EBP Q15125 3/20 0.39
SIGMAR1 Q99720 3/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
SLC22A2 O15244 1/20 0.36
SLC22A1 O15245 1/20 0.36
PGR P06401 1/20 0.36
THRB P10828 1/20 0.36
ADRB3 P13945 1/20 0.36
OPRK1 P41145 1/20 0.36
BLM P54132 1/20 0.36
PMP22 Q01453 1/20 0.36
KCNH2 Q12809 1/20 0.36
PDE3A Q14432 1/20 0.36
SLC47A1 Q96FL8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11472302 0.95 EBP (0.39) OPRM1DRD3CYP2D6DRD2DRD4
SCHEMBL11530730 0.92 CYP2D6 (0.56) OPRM1DRD3CYP2D6DRD2DRD4
SCHEMBL11532046 0.86 CYP2D6 (0.46) OPRM1DRD3CYP2D6DRD2DRD4
SCHEMBL11536775 0.85 EBP (0.50) OPRM1DRD3CYP2D6DRD2DRD4
SCHEMBL11535404 0.84 CYP2D6 (0.40) OPRM1DRD3CYP2D6DRD2DRD4
SCHEMBL11469619 0.84 CYP3A4 (0.34) OPRM1DRD3CYP2D6DRD2DRD4
SCHEMBL11479884 0.83 HRH3 (0.38) OPRM1DRD3CYP2D6DRD2DRD4
SCHEMBL11480207 0.82 KCNA3 (0.46) OPRM1CYP2D6CYP3A4KCNH2CHRM2
SCHEMBL11487964 0.81 KCNA3 (0.48) OPRM1CYP2D6CYP3A4KCNH2CHRM2
SCHEMBL10516752 0.81 TDP1 (0.44) OPRM1DRD3CYP2D6DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4217306-A ANTIARRHYTHMIA AGENTS G. D. SEARLE & CO. (US) 1980-08-12 US disclosed