SCHEMBL11535404

SCHEMBL11535404

CC(C)N(CCC(C#N)(CCN(C)C)c1ccc(F)cc1)C(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.40
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
OPRM1 P35372 1/20 0.40
DRD3 P35462 1/20 0.40
TAAR1 Q96RJ0 1/20 0.36
EBP Q15125 1/20 0.33
SIGMAR1 Q99720 1/20 0.33
CYP3A4 P08684 2/20 0.33
CASP1 P29466 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
SLC22A2 O15244 1/20 0.30
SLC22A1 O15245 1/20 0.30
PGR P06401 1/20 0.30
THRB P10828 1/20 0.30
ADRB3 P13945 1/20 0.30
OPRK1 P41145 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11536251 0.94 CASP1 (0.33) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11530730 0.86 CYP2D6 (0.56) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11470978 0.84 OPRM1 (0.48) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11534061 0.81 CASP1 (0.34) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11537461 0.80 KCNA3 (0.41) CYP2D6SIGMAR1SLC6A4
SCHEMBL11533486 0.80 ALDH1A1 (0.39) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11536775 0.80 EBP (0.50) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11532046 0.79 CYP2D6 (0.46) CYP2D6DRD2DRD4OPRM1DRD3
SCHEMBL11533529 0.78 TAAR1 (0.36) CYP2D6DRD2DRD4OPRM1DRD3
Hydrochloric Acid SCHEMBL10920199 0.77 SIGMAR1 (0.48) CYP2D6DRD2DRD4OPRM1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4153797-A α-Aryl-α, α-bis[ω- (disubstituted amino)alkyl]acetamides and related compounds G. D. SEARLE & CO. (US) 1979-05-08 US disclosed
US-4107205-A α-Aryl-α,α-bis[ω-(disubstituted amino)alkyl]acetamides and related compounds G. D. SEARLE & CO. (US) 1978-08-15 US disclosed