SCHEMBL11530730

SCHEMBL11530730

CC(C)N(CCC(C#N)(CCN(C)C)c1ccccc1)C(C)C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 3/20 0.56
OPRM1 P35372 3/20 0.56
DRD3 P35462 3/20 0.56
DRD2 P14416 2/20 0.56
DRD4 P21917 2/20 0.56
CYP3A4 P08684 2/20 0.47
EBP Q15125 3/20 0.44
SIGMAR1 Q99720 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
OPRK1 P41145 2/20 0.41
KCNH2 Q12809 2/20 0.41
SLC22A2 O15244 1/20 0.41
SLC22A1 O15245 1/20 0.41
PGR P06401 1/20 0.41
THRB P10828 1/20 0.41
ADRB3 P13945 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
PDE3A Q14432 1/20 0.41
SLC47A1 Q96FL8 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11532046 0.94 CYP2D6 (0.46) CYP2D6OPRM1DRD3DRD2DRD4
SCHEMBL11536775 0.93 EBP (0.50) CYP2D6OPRM1DRD3DRD2DRD4
SCHEMBL11470978 0.92 OPRM1 (0.48) CYP2D6OPRM1DRD3DRD2DRD4
SCHEMBL11537087 0.88 EBP (0.50) CYP2D6OPRM1DRD3DRD2DRD4
SCHEMBL11539556 0.87 SIGMAR1 (0.47) CYP2D6OPRM1DRD3DRD2DRD4
SCHEMBL11535404 0.86 CYP2D6 (0.40) CYP2D6OPRM1DRD3DRD2DRD4
SCHEMBL11532266 0.86 SIGMAR1 (0.43) CYP2D6OPRM1DRD3DRD2DRD4
SCHEMBL11472302 0.85 EBP (0.39) CYP2D6OPRM1DRD3DRD2DRD4
SCHEMBL10938259 0.82 CYP3A4 (0.47) CYP2D6OPRM1DRD3DRD2DRD4
SCHEMBL11481929 0.82 CYP3A4 (0.39) CYP2D6OPRM1DRD3DRD2DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4153797-A α-Aryl-α, α-bis[ω- (disubstituted amino)alkyl]acetamides and related compounds G. D. SEARLE & CO. (US) 1979-05-08 US disclosed
US-4107205-A α-Aryl-α,α-bis[ω-(disubstituted amino)alkyl]acetamides and related compounds G. D. SEARLE & CO. (US) 1978-08-15 US disclosed