SCHEMBL11486646

SCHEMBL11486646

O=C1C2=C(SCCS2)C(=O)N1c1ccc2ccc(O)nc2n1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
S100A4 P26447 1/20 0.32
PABPC1 P11940 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5201507 0.80 ALDH1A1 (0.40) ALDH1A1KMT2A
SCHEMBL11836641 0.79 ALDH1A1 (0.42) ALDH1A1NPSR1CRHBPCRHR2KMT2A
SCHEMBL11828982 0.79 ALDH1A1 (0.36) ALDH1A1NPSR1CRHBPCRHR2
SCHEMBL11849277 0.78 ALDH1A1 (0.44) ALDH1A1NPSR1CRHBPCRHR2S100A4
SCHEMBL11486146 0.76 CA12 (0.40)
SCHEMBL11833969 0.75
SCHEMBL11844709 0.70 ALDH1A1 (0.38) ALDH1A1NPSR1CRHBPCRHR2L3MBTL1
SCHEMBL11857335 0.70 ALDH1A1 (0.38) ALDH1A1NPSR1CRHBPCRHR2
SCHEMBL11260968 0.67 RECQL (0.34)
SCHEMBL12910406 0.66 PTPN22 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4220646-A TRANQUILIZERS, ANTICONVULSANTS, MUSCLE RELAXANTS, HYPNOTIC AGENTS RHONE-POULENC INDUSTRIES (FR) 1980-09-02 US disclosed
US-3966931-A TRANQUILIZERS, ANTICONVULSANTS, HYPNOSIS RHONE-POULENC S.A. (FR) 1976-06-29 US disclosed
US-3948917-A TRANQUILIZERS, ANTICONVULSANTS, DECONTRACTURANTS, HYPNOSIS RHONE-POULENC S.A. (FR) 1976-04-06 US disclosed