SCHEMBL11495147

SCHEMBL11495147

CCc1onc(C(=O)OCc2ccccc2)c1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
TDP1 Q9NUW8 4/20 0.45
KMT2A Q03164 4/20 0.45
SLC6A2 P23975 1/20 0.45
SLC6A3 Q01959 1/20 0.45
HTT P42858 2/20 0.43
PKM P14618 1/20 0.43
L3MBTL1 Q9Y468 4/20 0.43
TSHR P16473 3/20 0.43
CYP3A4 P08684 1/20 0.43
MAPK1 P28482 1/20 0.43
RAB9A P51151 5/20 0.42
MAPT P10636 4/20 0.42
ATM Q13315 2/20 0.42
STAT1 P42224 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MAOB P27338 1/20 0.42
ADORA2A P29274 1/20 0.42
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11496497 0.82 ALDH1A1 (0.45) ALDH1A1HTTTSHRKDM4E
SCHEMBL17409114 0.78 PPARG (0.44) ALDH1A1KMT2AHTTL3MBTL1TSHR
SCHEMBL25515307 0.74 HTT (0.46) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL23596007 0.73 TSHR (0.50) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL23596005 0.73 TDP1 (0.47) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL19035744 0.73 LMNA (0.45) ALDH1A1TDP1PKML3MBTL1TSHR
SCHEMBL15932081 0.73 KMT2A (0.46) ALDH1A1KMT2AHTTPKMTSHR
SCHEMBL2490988 0.73 TARBP2 (0.59) ALDH1A1TDP1KMT2ASLC6A2SLC6A3
SCHEMBL19167952 0.72 CA9 (0.47) ALDH1A1TDP1HTTL3MBTL1TSHR
SCHEMBL20031388 0.72 RAB9A (0.52) ALDH1A1TDP1KMT2ASLC6A2SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0012435-A2 Isoxazole derivatives, process for their preparation, medicines containing them and intermediates required in this process HOECHST AKTIENGESELLSCHAFT (DE) 1980-06-25 EP disclosed