SCHEMBL11517536

SCHEMBL11517536

Cc1noc(-c2ccccc2Cl)c1C(=O)Cl

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.52
GPBAR1 Q8TDU6 8/20 0.47
LMNA P02545 2/20 0.47
THRB P10828 1/20 0.46
ALDH1A1 P00352 1/20 0.45
NPC1 O15118 1/20 0.45
CYP2C19 P33261 2/20 0.45
PLAU P00749 1/20 0.44
ELANE P08246 1/20 0.44
EPAS1 Q99814 1/20 0.44
MAPT P10636 1/20 0.44
CYP3A4 P08684 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12543516 0.88 KMT2A (0.49) HSD17B10GPBAR1LMNATHRBALDH1A1
SCHEMBL30395754 0.88 KMT2A (0.49) HSD17B10GPBAR1LMNATHRBALDH1A1
SCHEMBL30576270 0.87 HSD17B10 (0.62) HSD17B10GPBAR1LMNATHRBALDH1A1
SCHEMBL11517946 0.84 ALDH1A1 (0.42) HSD17B10GPBAR1LMNATHRBALDH1A1
SCHEMBL11517887 0.82 POLB (0.47) GPBAR1LMNAALDH1A1NPC1MAPT
SCHEMBL30395634 0.82 ALDH1A1 (0.60) HSD17B10GPBAR1LMNAALDH1A1NPC1
SCHEMBL893014 0.80 PTGS1 (0.51) HSD17B10ALDH1A1MAPT
SCHEMBL11516385 0.79 GHSR (0.43) HSD17B10LMNAALDH1A1NPC1MAPT
SCHEMBL32679558 0.79 HSD17B10 (0.76) HSD17B10GPBAR1LMNAALDH1A1NPC1
SCHEMBL315858 0.79 HSD17B10 (0.76) HSD17B10GPBAR1LMNAALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106316975-A Amide compound and application thereof as TGR5 agonist 山东轩竹医药科技有限公司 2017-01-11 CN disclosed
US-4155905-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1979-05-22 US disclosed
US-4077967-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1978-03-07 US disclosed
US-4061629-A 6-Amino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4061851-A 7-Amino-7-arylthio cephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4029669-A 6-Benzalimino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-06-14 US disclosed
US-4026886-A 7-Acyl-7-arylthiocephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-05-31 US disclosed
US-3965093-A 6-Arylthio penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1976-06-22 US disclosed
US-3954744-A ANTIBACTERIAL E. R. SQUIBB & SONS, INC. (US) 1976-05-04 US disclosed