SCHEMBL11518482

SCHEMBL11518482

Cc1ccc(-c2cncc(O)n2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.47
CYP11B2 P19099 2/20 0.47
ENPP3 O14638 1/20 0.44
ENPP1 P22413 1/20 0.44
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
METAP2 P50579 1/20 0.41
METAP1 P53582 1/20 0.41
FYN P06241 2/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
KDM4E B2RXH2 3/20 0.40
SCN2A Q99250 1/20 0.39
SCN10A Q9Y5Y9 1/20 0.39
CHEK1 O14757 2/20 0.39
ALDH1A1 P00352 2/20 0.39
MITF O75030 1/20 0.39
KDM5A P29375 1/20 0.39
KDM5C P41229 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4910639 0.85 CYP11B1 (0.59) CYP11B1CYP11B2ENPP3ENPP1MEN1
SCHEMBL11679588 0.80 RAB9A (0.46) MEN1KMT2AMETAP2NPC1RAB9A
SCHEMBL18662151 0.80 SCN10A (0.39) CYP11B1CYP11B2FYNNPC1RAB9A
SCHEMBL23121272 0.80 FYN (0.47) MEN1KMT2AMETAP2FYNNPC1
SCHEMBL5647023 0.80 CYP11B1 (0.47) CYP11B1CYP11B2ENPP3ENPP1MEN1
SCHEMBL18850044 0.79 CYP11B1 (0.50) CYP11B1CYP11B2ENPP3ENPP1MEN1
SCHEMBL11516493 0.79 CHEK1 (0.46) CYP11B1CYP11B2MEN1KMT2ANPC1
SCHEMBL13264053 0.78 MEN1 (0.56) CYP11B1CYP11B2MEN1KMT2ANPC1
SCHEMBL4901225 0.76 CYP11B2 (0.49) CYP11B1CYP11B2ENPP3ENPP1MEN1
SCHEMBL31301361 0.74 SCN10A (0.51) CYP11B1CYP11B2SMN1; SMN2SCN2ASCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4162319-A ANTHELMINTICS, PSYCHOTROPIC, CNS, HYPOGLYCOMIC AGENTS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1979-07-24 US disclosed
US-4120961-A ANTIHELMINTICS, CNS ACITVITY E. MERCK (DE) 1978-10-17 US disclosed
US-4051243-A RING SUBSTITUTED PYRAZINO-ISOQUINOLINE DERIVATIVES AND THEIR PREPARATION MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-09-27 US disclosed