SCHEMBL11520591

SCHEMBL11520591

Cc1ccc(-c2onc(C)c2C(=O)Cl)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 5/20 0.44
NPC1 O15118 4/20 0.44
RAB9A P51151 4/20 0.44
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
ALDH1A1 P00352 3/20 0.44
IP6K1 Q92551 2/20 0.44
IP6K3 Q96PC2 2/20 0.44
IP6K2 Q9UHH9 2/20 0.44
KDM4E B2RXH2 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
NPSR1 Q6W5P4 2/20 0.44
NR1I2 O75469 1/20 0.44
MAPT P10636 3/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
USP2 O75604 1/20 0.40
HPGD P15428 1/20 0.39
PTK2B Q14289 1/20 0.39
LMNA P02545 2/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11518747 0.89 MAPT (0.51) POLBNPC1RAB9AKMT2AMEN1
SCHEMBL1784 0.87 ALDH1A1 (0.40) POLBNPC1RAB9AKMT2AMEN1
SCHEMBL893014 0.87 PTGS1 (0.51) KMT2AMEN1ALDH1A1IP6K1IP6K3
SCHEMBL15280716 0.85 RAB9A (0.52) POLBNPC1RAB9AKMT2AMEN1
SCHEMBL14789796 0.83 RAB9A (0.51) POLBNPC1RAB9AKMT2AMEN1
SCHEMBL14789793 0.80 HTT (0.57) POLBNPC1RAB9AKMT2AMEN1
SCHEMBL4336589 0.75 MAPT (0.51) POLBNPC1RAB9AKMT2AMEN1
SCHEMBL11515850 0.73 GPBAR1 (0.59) POLBKMT2AMEN1SMN1; SMN2USP2
SCHEMBL22467553 0.73 ALDH1A1 (0.46) POLBNPC1RAB9AKMT2AMEN1
SCHEMBL13508 0.73 PTGS1 (0.51) KMT2AMEN1ALDH1A1IP6K1IP6K3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4155905-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1979-05-22 US disclosed
US-4077967-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1978-03-07 US disclosed
US-4061629-A 6-Amino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4061851-A 7-Amino-7-arylthio cephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4029669-A 6-Benzalimino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-06-14 US disclosed
US-4026886-A 7-Acyl-7-arylthiocephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-05-31 US disclosed
US-3965093-A 6-Arylthio penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1976-06-22 US disclosed
US-3954744-A ANTIBACTERIAL E. R. SQUIBB & SONS, INC. (US) 1976-05-04 US disclosed