SCHEMBL11520754

SCHEMBL11520754

Cc1onc(-c2ccccc2[N+](=O)[O-])c1C(=O)Cl

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.59
HSD17B10 Q99714 1/20 0.50
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA4 P22748 1/20 0.47
CA7 P43166 1/20 0.47
GPBAR1 Q8TDU6 3/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPT P10636 2/20 0.45
LMNA P02545 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
GAA P10253 1/20 0.45
TNF P01375 1/20 0.44
NOD2 Q9HC29 1/20 0.44
NOD1 Q9Y239 1/20 0.44
NPC1 O15118 1/20 0.44
CYP2C19 P33261 1/20 0.44
PLAU P00749 1/20 0.43
ELANE P08246 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29059028 0.88 GHSR (0.60) GHSRHSD17B10CA1CA2CA4
SCHEMBL11516385 0.82 GHSR (0.43) GHSRHSD17B10CA1CA2CA4
SCHEMBL32679558 0.79 HSD17B10 (0.76) HSD17B10GPBAR1ALDH1A1MAPTLMNA
SCHEMBL315858 0.79 HSD17B10 (0.76) HSD17B10GPBAR1ALDH1A1MAPTLMNA
SCHEMBL892042 0.77 KMT2A (0.71) GPBAR1ALDH1A1LMNAMEN1KMT2A
SCHEMBL11517059 0.77 MEN1 (0.55) GPBAR1ALDH1A1LMNAMEN1KMT2A
SCHEMBL11518678 0.76 GPBAR1 (0.64) GHSRHSD17B10GPBAR1ALDH1A1MAPT
SCHEMBL3632594 0.75 GHSR (1.00) GHSRCA1CA2CA4CA7
SCHEMBL29058691 0.73 EPAS1 (0.74) GHSRCA1CA2CA4CA7
SCHEMBL10473335 0.72 TDP1 (0.47) GHSRHSD17B10ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4155905-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1979-05-22 US disclosed
US-4077967-A 6-Substituted penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1978-03-07 US disclosed
US-4061629-A 6-Amino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4061851-A 7-Amino-7-arylthio cephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-12-06 US disclosed
US-4029669-A 6-Benzalimino-6-arylthio penicillanic acids and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1977-06-14 US disclosed
US-4026886-A 7-Acyl-7-arylthiocephalosporins E. R. SQUIBB & SONS, INC. (US) 1977-05-31 US disclosed
US-3965093-A 6-Arylthio penicillanic acid and derivatives thereof E. R. SQUIBB & SONS, INC. (US) 1976-06-22 US disclosed
US-3954744-A ANTIBACTERIAL E. R. SQUIBB & SONS, INC. (US) 1976-05-04 US disclosed