SCHEMBL11523852

SCHEMBL11523852

Cc1cccc(C)c1C(=O)NC(=O)Nc1cnc(-c2cccc(C#N)c2)cn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 2/20 0.45
PRKDC P78527 1/20 0.45
GRM5 P41594 2/20 0.44
ADORA2A P29274 2/20 0.42
ADORA1 P30542 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPK1 P28482 3/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
HSD17B10 Q99714 2/20 0.40
ALDH1A1 P00352 2/20 0.40
CLK4 Q9HAZ1 1/20 0.40
CTSA P10619 1/20 0.40
HDAC2 Q92769 1/20 0.40
LRRK2 Q5S007 1/20 0.40
MAPK14 Q16539 1/20 0.40
KDM4E B2RXH2 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11521631 0.84 WNT3A (0.45) NPC1RAB9ASMN1; SMN2MAPTSTIM1
SCHEMBL11521495 0.78 PIK3CA (0.42) GRM5NPC1RAB9ASMN1; SMN2MAPK1
SCHEMBL11527118 0.73 STIM1 (0.42) ATRPRKDCNPC1RAB9ASMN1; SMN2
SCHEMBL11604630 0.71 RAB9A (0.48) NPC1RAB9AKDM4EMAPT
SCHEMBL11521003 0.70 KMO (0.45) NPC1RAB9AMAPT
SCHEMBL11522661 0.70 IL2 (0.42) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL11523521 0.70 PDE10A (0.38) NPC1RAB9ASMN1; SMN2MAPK1CYP1A2
SCHEMBL11524371 0.69 MAPT (0.45) HSD17B10ALDH1A1KDM4EMAPTHPGD
SCHEMBL11521149 0.69 NPC1 (0.46) NPC1RAB9ASMN1; SMN2MAPTHPGD
SCHEMBL11526321 0.69 STIM1 (0.42) NPC1RAB9AALDH1A1MAPTSTIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4160834-A INSECTICIDES ELI LILLY AND COMPANY (US) 1979-07-10 US disclosed
US-4083977-A Novel insecticidal 1-(substituted benzoyl)-3-(substituted pyrazinyl)ureas ELI LILLY AND COMPANY (US) 1978-04-11 US disclosed