SCHEMBL11528320

SCHEMBL11528320

CCOC(=O)c1cc(N(C)C)ncn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
GABRA1 P14867 7/20 0.43
GABRG2 P18507 7/20 0.43
GABRB3 P28472 7/20 0.43
GABRA5 P31644 7/20 0.43
GABRA3 P34903 7/20 0.43
GABRA2 P47869 7/20 0.43
GABRA4 P48169 7/20 0.43
GABRA6 Q16445 7/20 0.43
GABRP O00591 6/20 0.43
GABRD O14764 6/20 0.43
GABRB1 P18505 6/20 0.43
GABRB2 P47870 6/20 0.43
GABRE P78334 6/20 0.43
GABRG1 Q8N1C3 6/20 0.43
GABRG3 Q99928 6/20 0.43
GABRQ Q9UN88 6/20 0.43
ALDH1A1 P00352 4/20 0.41
NPC1 O15118 3/20 0.41
MAPT P10636 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11530632 0.81 TP53 (0.34) CYP1A2ALDH1A1NPC1KDM4ESMN1; SMN2
SCHEMBL3036654 0.80 S1PR1 (0.56) ALDH1A1JAK3
SCHEMBL10228362 0.80 CYP1A2 (0.50) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL294157 0.78 CYP1A2 (0.49) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL549184 0.77 CYP1A2 (0.47) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL13472450 0.77 ALDH1A1 (0.47) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL8328525 0.75 ALDH1A1 (0.50) CYP1A2ALDH1A1MAPTKDM4EHSD17B10
SCHEMBL17550606 0.75 POLB (0.46) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL25276749 0.73 CYP1A2 (0.44) CYP1A2GABRA1GABRG2GABRB3GABRA5
SCHEMBL29537507 0.73 CYP1A2 (0.44) CYP1A2GABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4144339-A TREATMENT OF BILHARZIASIS RHONE-POULENC INDUSTRIES (FR) 1979-03-13 US disclosed
US-4138487-A NEMATOCIDES RHONE-POULENC INDUSTRIES (FR) 1979-02-06 US disclosed
US-4110450-A BILHARZIASIS RHONE-POULENC INDUSTRIES (FR) 1978-08-29 US disclosed