SCHEMBL11530632

SCHEMBL11530632

CCOC(=O)C(C)C(=O)c1cc(N(C)C)ncn1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.34
KDM4E B2RXH2 1/20 0.34
KCNH2 Q12809 1/20 0.34
S1PR1 P21453 5/20 0.33
HTT P42858 2/20 0.33
S1PR3 Q99500 1/20 0.33
LMNA P02545 1/20 0.33
ALDH1A1 P00352 3/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
ELOVL1 Q9BW60 1/20 0.32
NPC1 O15118 1/20 0.32
ALOX15 P16050 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11529393 0.76 HTR1A (0.37) TP53HTTLMNAALDH1A1CYP1A2
SCHEMBL3567261 0.72 P2RX7 (0.45) ALDH1A1CYP1A2MEN1KMT2ASMN1; SMN2
SCHEMBL11529183 0.70 ALDH1A1 (0.49) KDM4EHTTLMNAALDH1A1HSD17B10
SCHEMBL11530272 0.69 POLB (0.49) KDM4EHTTLMNAALDH1A1HSD17B10
SCHEMBL11529414 0.68 SMN1; SMN2 (0.48) TP53KDM4EHTTLMNAALDH1A1
SCHEMBL27196361 0.68 GSK3B (0.51) KDM4EHTTLMNAALDH1A1CYP1A2
SCHEMBL29852720 0.67 CA12 (0.36) KDM4EKCNH2S1PR1S1PR3LMNA
SCHEMBL11528581 0.66 CYP1A2 (0.38) KDM4EHTTLMNAALDH1A1CYP1A2
SCHEMBL11529854 0.65 CYP2C9 (0.42) TP53KDM4ELMNAALDH1A1CYP1A2
SCHEMBL3405792 0.65 HTT (0.43) HTTLMNAALDH1A1CYP1A2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4144339-A TREATMENT OF BILHARZIASIS RHONE-POULENC INDUSTRIES (FR) 1979-03-13 US disclosed
US-4138487-A NEMATOCIDES RHONE-POULENC INDUSTRIES (FR) 1979-02-06 US disclosed
US-4110450-A BILHARZIASIS RHONE-POULENC INDUSTRIES (FR) 1978-08-29 US disclosed