SCHEMBL8328525

SCHEMBL8328525

CN(C)c1cc(C(=O)O)ncn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
KDM4E B2RXH2 3/20 0.50
KMO O15229 16/20 0.46
HSD17B10 Q99714 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C19 P33261 1/20 0.39
KDM6B O15054 1/20 0.38
TET3 O43151 1/20 0.38
KDM4A O75164 1/20 0.38
BBOX1 O75936 1/20 0.38
MAPT P10636 1/20 0.38
KDM5A P29375 1/20 0.38
KDM5C P41229 1/20 0.38
ASPH Q12797 1/20 0.38
KDM4D Q6B0I6 1/20 0.38
TET2 Q6N021 1/20 0.38
ALKBH5 Q6P6C2 1/20 0.38
KDM7A Q6ZMT4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL71141 0.78 KMO (0.59) ALDH1A1KDM4EKMOKDM6BTET3
SCHEMBL3233039 0.77 KDM4E (0.46) ALDH1A1KDM4EHSD17B10CYP1A2CYP3A4
SCHEMBL2771569 0.76 S1PR1 (0.62) KMO
SCHEMBL21442941 0.76 KMO (0.38) ALDH1A1KDM4EKMO
SCHEMBL11528320 0.75 CYP1A2 (0.45) ALDH1A1KDM4EHSD17B10CYP1A2MAPT
Hydrochloric Acid SCHEMBL3272233 0.75 KMO (0.57) ALDH1A1KDM4EKMOKDM6BTET3
Fluoride SCHEMBL21173953 0.75 KMO (0.57) ALDH1A1KDM4EKMOKDM6BTET3
Hydrochloric Acid SCHEMBL3272369 0.75 KMO (0.57) ALDH1A1KDM4EKMOKDM6BTET3
SCHEMBL7717522 0.75 CYP1A2 (0.50) ALDH1A1HSD17B10CYP1A2CYP3A4CYP2D6
SCHEMBL29852720 0.73 CA12 (0.36) ALDH1A1KDM4EKMO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948495-A1 ARYL AND HETEROARYL SUBSTITUTED FUSED PYRROLE ANTIINFLAMMATORY AGENTS Amgen Inc., (US) 1999-10-13 EP disclosed
WO-1998022457-A9 ARYL AND HETEROARYL SUBSTITUTED FUSED PYRROLE ANTIINFLAMMATORY AGENTS 1998-08-20 WO disclosed
WO-1998022457-A1 ARYL AND HETEROARYL SUBSTITUTED FUSED PYRROLE ANTIINFLAMMATORY AGENTS AMGEN INC. (US) 1998-05-28 WO disclosed
US-4144339-A TREATMENT OF BILHARZIASIS RHONE-POULENC INDUSTRIES (FR) 1979-03-13 US disclosed
US-4138487-A NEMATOCIDES RHONE-POULENC INDUSTRIES (FR) 1979-02-06 US disclosed
US-4110450-A BILHARZIASIS RHONE-POULENC INDUSTRIES (FR) 1978-08-29 US disclosed