SCHEMBL11528657

SCHEMBL11528657

O=C(O)CCCc1nn[nH]c1S.[NaH].[NaH]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.35
MAPK1 P28482 1/20 0.35
ADRA1A P35348 1/20 0.35
HDAC4 P56524 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HDAC1 Q13547 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
TBXAS1 P24557 9/20 0.34
LMNA P02545 2/20 0.33
SLC22A6 Q4U2R8 1/20 0.33
ALDH1A1 P00352 1/20 0.33
FOLH1 Q04609 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11529642 0.98 HDAC3 (0.36) HDAC3MAPK1ADRA1AHDAC4SLC6A3
SCHEMBL11529545 0.89 ALDH1A1 (0.41) HDAC6ALDH1A1HSD17B10
SCHEMBL11529126 0.87 ALDH1A1 (0.42) HDAC6ALDH1A1HSD17B10
SCHEMBL11535089 0.78 GABRR1 (0.35) LMNA
SCHEMBL11530172 0.74 BLM (0.38) TBXAS1LMNA
SCHEMBL11531740 0.71 ALDH1A1 (0.41) SMN1; SMN2LMNAALDH1A1TSHRHSD17B10
SCHEMBL11529284 0.69 ALDH1A1 (0.42) MAPK1SMN1; SMN2LMNAALDH1A1TSHR
SCHEMBL8627216 0.64 HDAC3 (0.41) HDAC3MAPK1ADRA1AHDAC4SLC6A3
SCHEMBL11526838 0.63 HCAR2 (0.32)
SCHEMBL11528231 0.61

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4142046-A BACTERICIDES, 7-AMINO-CEPHALOSPORINS SMITHKLINE CORPORATION (US) 1979-02-27 US disclosed
US-4060610-A Pharmaceutical compositions comprising 7-acyl-3-(substituted triazolyl thiomethyl)-cephalosporins and methods of treating bacterial infections SMITHKLINE CORPORATION (US) 1977-11-29 US disclosed
US-3989694-A ANTIBACTERIAL SMITHKLINE CORPORATION (US) 1976-11-02 US disclosed