SCHEMBL11529545

SCHEMBL11529545

O=C(O)CCc1nn[nH]c1S.[NaH].[NaH]

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
HDAC6 Q9UBN7 3/20 0.32
KEAP1 Q14145 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KDM4E B2RXH2 1/20 0.30
TP53 P04637 1/20 0.30
POLB P06746 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11529126 0.98 ALDH1A1 (0.42) ALDH1A1HDAC6KEAP1L3MBTL1KDM4E
SCHEMBL11528657 0.89 HDAC3 (0.35) ALDH1A1HDAC6HSD17B10
SCHEMBL11535089 0.81 GABRR1 (0.35)
SCHEMBL11531740 0.77 ALDH1A1 (0.41) ALDH1A1L3MBTL1KDM4EHSD17B10
SCHEMBL11529284 0.75 ALDH1A1 (0.42) ALDH1A1L3MBTL1KDM4EHSD17B10
SCHEMBL11530172 0.70 BLM (0.38)
SCHEMBL11526838 0.66 HCAR2 (0.32)
SCHEMBL11528231 0.63
SCHEMBL2704416 0.63 CHRM1 (0.39) ALDH1A1KEAP1KDM4E
SCHEMBL8631052 0.61 KEAP1 (0.37) ALDH1A1KEAP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4142046-A BACTERICIDES, 7-AMINO-CEPHALOSPORINS SMITHKLINE CORPORATION (US) 1979-02-27 US disclosed
US-4060610-A Pharmaceutical compositions comprising 7-acyl-3-(substituted triazolyl thiomethyl)-cephalosporins and methods of treating bacterial infections SMITHKLINE CORPORATION (US) 1977-11-29 US disclosed
US-3989694-A ANTIBACTERIAL SMITHKLINE CORPORATION (US) 1976-11-02 US disclosed