SCHEMBL11530952

SCHEMBL11530952

CCC(=O)C(Cc1ccc(/C=C/c2ccc(OC)cc2Cl)cc1Cl)C(=O)CC

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 2/20 0.40
RELA Q04206 1/20 0.40
CYP1A1 P04798 5/20 0.38
CYP1B1 Q16678 5/20 0.38
CYP1A2 P05177 4/20 0.38
BACE1 P56817 3/20 0.37
NR1H4 Q96RI1 4/20 0.36
APP P05067 1/20 0.36
MAPT P10636 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CYP19A1 P11511 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11530957 1.00 NFE2L2 (0.40) NFE2L2RELACYP1A1CYP1B1CYP1A2
SCHEMBL11527964 0.87 NFE2L2 (0.44) NFE2L2RELACYP1A1CYP1B1CYP1A2
SCHEMBL11527960 0.87 NFE2L2 (0.44) NFE2L2RELACYP1A1CYP1B1CYP1A2
SCHEMBL11306176 0.86 LDHA (0.41)
SCHEMBL11530709 0.78 RELA (0.48) NFE2L2RELACYP1A1CYP1B1CYP1A2
SCHEMBL11530716 0.78 RELA (0.48) NFE2L2RELACYP1A1CYP1B1CYP1A2
SCHEMBL11457464 0.75 LDHA (0.48)
SCHEMBL11527142 0.72 HTR2A (0.34)
SCHEMBL11525535 0.72 RELA (0.53) NFE2L2RELACYP1A1CYP1B1CYP1A2
SCHEMBL11525531 0.72 RELA (0.53) NFE2L2RELACYP1A1CYP1B1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4153719-A Aromatic diketones STERLING DRUG INC. (US) 1979-05-08 US claimed
US-4153719-A Aromatic diketones STERLING DRUG INC. (US) 1979-05-08 US disclosed