SCHEMBL11535640

SCHEMBL11535640

Clc1ccc(C(c2ccccc2)c2ccncc2)cc1

nearest known ligand 0.83

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 0.83
SLC6A2 P23975 3/20 0.75
SLC6A4 P31645 3/20 0.75
SLC6A3 Q01959 3/20 0.75
CFTR P13569 1/20 0.50
GOPC Q9HD26 1/20 0.50
AKT1 P31749 2/20 0.47
IDO1 P14902 2/20 0.47
TDO2 P48775 2/20 0.47
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
SLC6A9 P48067 1/20 0.44
S1PR1 P21453 1/20 0.44
S1PR3 Q99500 1/20 0.44
CNR1 P21554 1/20 0.43
PRCP P42785 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11538836 0.91 CYP19A1 (1.00) CYP19A1SLC6A2SLC6A4SLC6A3AKT1
SCHEMBL733008 0.87 SLC6A3 (1.00) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL673181 0.87 CYP19A1 (0.59) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL3695767 0.87 CYP19A1 (0.59) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
Ammonia Solution, Strong SCHEMBL5999715 0.84 SLC6A3 (0.95) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL22388390 0.80 CYP1A2 (0.64) CYP19A1SLC6A2SLC6A4SLC6A3AKT1
SCHEMBL8176557 0.80 CYP19A1 (0.85) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL14393365 0.79 SLC6A2 (0.75) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL10038666 0.79 SLC6A2 (0.75) CYP19A1SLC6A2SLC6A4SLC6A3CFTR
SCHEMBL6501455 0.78 CYP19A1 (0.68) CYP19A1SLC6A2SLC6A4SLC6A3AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4180660-A CONTAINING FORMYL SUBSTITUTED PYRROLE GROUP YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 1979-12-25 US disclosed
US-4148998-A ANTIBIOTICS YEDA RESEARCH AND DEVELOPMENT CO., LTD. (IL) 1979-04-10 US disclosed
US-4138488-A Diphenylmethyl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-06 US disclosed
US-4122260-A CONTAINING FORMYL SUBSTITUTED PYRROLE, ANTIBIOTICS YEDA RESEARCH AND DEVELOPMENT CO., LTD. (IL) 1978-10-24 US disclosed