SCHEMBL11536196

SCHEMBL11536196

N#CCOC(=O)c1ccc(C(c2ccccc2)(c2ccccc2)c2ccc(Cl)cc2)cn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
KMT2A Q03164 4/20 0.36
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35
L3MBTL1 Q9Y468 3/20 0.34
MAPT P10636 3/20 0.34
RXFP1 Q9HBX9 1/20 0.34
AGTR1 P30556 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
RECQL P46063 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 3/20 0.34
POLB P06746 1/20 0.34
GABRA2 P47869 2/20 0.33
LTC4S Q16873 2/20 0.33
EGLN1 Q9GZT9 1/20 0.33
P4HTM Q9NXG6 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11536417 0.95 KMT2A (0.38) ALDH1A1KMT2AMAPTCYP1A2CYP2C19
SCHEMBL11534109 0.94 ALDH1A1 (0.38) ALDH1A1KMT2AKDM4EPKML3MBTL1
SCHEMBL11538505 0.89 GABRA1 (0.40) ALDH1A1KMT2AKDM4EPKMMAPT
SCHEMBL11536777 0.88 ALDH1A1 (0.39) ALDH1A1KDM4EPKMMAPTRXFP1
SCHEMBL11536526 0.88 KMT2A (0.41) ALDH1A1KMT2AKDM4EPKML3MBTL1
SCHEMBL11534104 0.88 MAPT (0.36) ALDH1A1KDM4EPKML3MBTL1MAPT
SCHEMBL11535434 0.88 ALDH1A1 (0.38) ALDH1A1KMT2AKDM4EPKML3MBTL1
SCHEMBL11537930 0.86 ALDH1A1 (0.38) ALDH1A1KDM4EMAPTRXFP1CYP1A2
SCHEMBL11534846 0.84 ALDH1A1 (0.39) ALDH1A1KDM4EMAPTRXFP1SMN1; SMN2
SCHEMBL11542791 0.84 MEN1 (0.39) ALDH1A1KMT2AKDM4EPKML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139625-A 5-(Substituted triphenylmethyl)picolinamides and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-13 US disclosed
US-4133887-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-01-09 US disclosed
US-4127662-A ANTIACNE SCHERING CORPORATION (US) 1978-11-28 US disclosed
US-4123433-A ANTIACNE AGENTS SCHERING CORPORATION (US) 1978-10-31 US disclosed
US-4044140-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1977-08-23 US disclosed