SCHEMBL11537005

SCHEMBL11537005

Sc1nnc(C2CC2)n1-c1ccccc1Cl

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCAR1 Q9BXC0 1/20 0.47
TNKS2 Q9H2K2 4/20 0.41
NPSR1 Q6W5P4 1/20 0.39
AVPR1A P37288 4/20 0.39
TNKS O95271 1/20 0.37
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
HTT P42858 1/20 0.35
HSD17B10 Q99714 1/20 0.35
NOTUM Q6P988 2/20 0.35
ADRB1 P08588 1/20 0.34
GRM2 Q14416 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11538651 0.83 GRM2 (0.37) HCAR1AVPR1AALDH1A1ALOX15HTT
SCHEMBL21045356 0.77 HTT (0.51) AVPR1AALDH1A1ALOX15HTTHSD17B10
SCHEMBL11920145 0.77 SMN1; SMN2 (0.53) NPSR1HTT
SCHEMBL12892262 0.74 AVPR1A (0.45) AVPR1AALDH1A1ALOX15HTTHSD17B10
SCHEMBL5098675 0.74 HSD11B1 (0.41) HCAR1TNKS2NPSR1AVPR1ATNKS
SCHEMBL11538155 0.73 TNKS (0.42) HCAR1TNKS2TNKSALDH1A1NOTUM
SCHEMBL14112938 0.71 HSD11B1 (0.51) ALDH1A1ALOX15HSD17B10
SCHEMBL2640557 0.71 TNKS (0.48) TNKS2NPSR1TNKSALDH1A1ALOX15
SCHEMBL15790773 0.70 KCNN4 (0.47) HCAR1ALDH1A1NOTUM
SCHEMBL5334498 0.70 ALDH1A1 (0.45) NPSR1AVPR1AALDH1A1ALOX15HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4134914-A 1-Acyl-4-substituted phenyl thiosemicarbazides ELI LILLY AND COMPANY (US) 1979-01-16 US disclosed
US-4082762-A 4-(2-HALOPHENYL)-1,2,4-TRIAZOLE-3-THIOL COMPOUNDS ELI LILLY AND COMPANY (US) 1978-04-04 US disclosed
US-3937713-A Process for the preparation of s-triazolo[3,4-b]benzothiazoles ELI LILLY AND COMPANY (US) 1976-02-10 US disclosed