SCHEMBL11537872

SCHEMBL11537872

CCN(CC)CCn1c2c(c3ccccc31)CCS(=O)(=O)CCC2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.50
HRH1 P35367 2/20 0.50
CHRM2 P08172 1/20 0.50
HTR1A P08908 1/20 0.50
CHRM5 P08912 1/20 0.50
ADRA2A P08913 1/20 0.50
DRD2 P14416 1/20 0.50
ADRA2B P18089 1/20 0.50
ADRA2C P18825 1/20 0.50
CHRM3 P20309 1/20 0.50
DRD4 P21917 1/20 0.50
HRH2 P25021 1/20 0.50
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
AVPR2 P30518 1/20 0.50
ADRA1A P35348 1/20 0.50
DRD3 P35462 1/20 0.50
OPRK1 P41145 1/20 0.50
HTR2B P41595 1/20 0.50
HTR5A P47898 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11530224 0.88 CHRM2 (0.61) SLC6A2HRH1CHRM2HTR1ACHRM5
SCHEMBL11531885 0.84 CHRM2 (0.72) SLC6A2HRH1CHRM2HTR1ACHRM5
SCHEMBL25818911 0.71 HTR6 (0.85) SLC6A2HRH1CHRM2HTR1ACHRM5
SCHEMBL2334457 0.71 POLB (0.63) SLC6A2HRH1KDM4EALDH1A1TSHR
SCHEMBL18457140 0.70 CA1 (0.67) SLC6A2HRH1CHRM2HTR1ACHRM5
SCHEMBL11534971 0.70 HRH1 (0.52) SLC6A2HRH1CHRM2HTR1ACHRM5
Ammonia Solution, Strong SCHEMBL905721 0.69 CA1 (0.63) SLC6A2HRH1CHRM2HTR1ACHRM5
SCHEMBL10703956 0.69 SLC6A4 (0.78) SLC6A2HRH1KDM4EALDH1A1HIF1A
SCHEMBL1459437 0.67 CA1 (0.71) SLC6A2HRH1CHRM2HTR1ACHRM5
SCHEMBL30184445 0.67 CA1 (0.71) SLC6A2HRH1CHRM2HTR1ACHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4144349-A N,N-dimethyl-1,2,4,5,6,7-hexahydrothiocino[5,4-b]-indole-7-propanamine-3,3-dioxides and related thiocines WARNER-LAMBERT COMPANY (US) 1979-03-13 US claimed
US-4144349-A N,N-dimethyl-1,2,4,5,6,7-hexahydrothiocino[5,4-b]-indole-7-propanamine-3,3-dioxides and related thiocines WARNER-LAMBERT COMPANY (US) 1979-03-13 US disclosed