SCHEMBL11530224

SCHEMBL11530224

CN(C)CCn1c2c(c3ccccc31)CCS(=O)(=O)CCC2

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 2/20 0.61
HTR1A P08908 2/20 0.61
ADRA2A P08913 2/20 0.61
SLC6A2 P23975 2/20 0.61
ADRA1A P35348 2/20 0.61
DRD3 P35462 2/20 0.61
KCNH2 Q12809 2/20 0.61
HRH1 P35367 2/20 0.61
HTR6 P50406 2/20 0.61
CHRM5 P08912 1/20 0.61
DRD2 P14416 1/20 0.61
ADRA2B P18089 1/20 0.61
ADRA2C P18825 1/20 0.61
CHRM3 P20309 1/20 0.61
DRD4 P21917 1/20 0.61
HRH2 P25021 1/20 0.61
HTR2A P28223 1/20 0.61
HTR2C P28335 1/20 0.61
AVPR2 P30518 1/20 0.61
OPRK1 P41145 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11531885 0.93 CHRM2 (0.72) CHRM2HTR1AADRA2ASLC6A2ADRA1A
SCHEMBL11537872 0.88 SLC6A2 (0.50) CHRM2HTR1AADRA2ASLC6A2ADRA1A
SCHEMBL25818911 0.83 HTR6 (0.85) CHRM2HTR1AADRA2ASLC6A2ADRA1A
SCHEMBL11533022 0.78 HTR6 (0.64) CHRM2HTR1AADRA2ASLC6A2ADRA1A
SCHEMBL11534971 0.78 HRH1 (0.52) CHRM2HTR1AADRA2ASLC6A2ADRA1A
SCHEMBL11891460 0.76 HTR6 (1.00) CHRM2HTR1AADRA2ASLC6A2ADRA1A
Iprindole SCHEMBL49509 0.76 HTR6 (1.00) CHRM2HTR1AADRA2ASLC6A2ADRA1A
Iprindole SCHEMBL29407410 0.76 HTR6 (1.00) CHRM2HTR1AADRA2ASLC6A2ADRA1A
Iprindole SCHEMBL5705755 0.75 HTR6 (0.97) CHRM2HTR1AADRA2ASLC6A2ADRA1A
SCHEMBL7412035 0.72 HTR6 (0.55) CHRM2HTR1AADRA2ASLC6A2ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4144349-A N,N-dimethyl-1,2,4,5,6,7-hexahydrothiocino[5,4-b]-indole-7-propanamine-3,3-dioxides and related thiocines WARNER-LAMBERT COMPANY (US) 1979-03-13 US claimed
US-4144349-A N,N-dimethyl-1,2,4,5,6,7-hexahydrothiocino[5,4-b]-indole-7-propanamine-3,3-dioxides and related thiocines WARNER-LAMBERT COMPANY (US) 1979-03-13 US disclosed