SCHEMBL11537892

SCHEMBL11537892

COc1ccc(C(c2ccccc2)(c2ccccc2)c2ccc(Br)nc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 8/20 0.41
KCNH2 Q12809 1/20 0.41
CA4 P22748 1/20 0.39
LTA4H P09960 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
RAB9A P51151 3/20 0.38
NPC1 O15118 2/20 0.38
AHR P35869 1/20 0.38
SCN2A Q99250 1/20 0.37
MAPT P10636 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LMNA P02545 1/20 0.36
TRPA1 O75762 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11534894 0.87 NPC1 (0.33) RAB9ANPC1ALDH1A1SMN1; SMN2
SCHEMBL11534166 0.82 TSHR (0.38) KIF11MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL28067932 0.81 CA4 (0.59) KIF11KCNH2CA4LTA4HRAB9A
SCHEMBL10112758 0.81 CA4 (0.59) KIF11KCNH2CA4LTA4HRAB9A
SCHEMBL11533455 0.80 NPC1 (0.44) KIF11MEN1KMT2ARAB9ANPC1
SCHEMBL11539601 0.79 NPC1 (0.40) KIF11KCNH2CA4LTA4HMEN1
SCHEMBL11535711 0.79 CYP19A1 (0.40) KIF11MEN1KMT2ARAB9ANPC1
SCHEMBL11541379 0.79 ALDH1A1 (0.48) KIF11KMT2ARAB9ANPC1SCN2A
SCHEMBL11535231 0.79 KCNN4 (0.39) KIF11KCNH2MEN1KMT2ARAB9A
SCHEMBL11538266 0.78 P4HTM (0.51) KIF11RAB9ANPC1MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139625-A 5-(Substituted triphenylmethyl)picolinamides and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-13 US disclosed
US-4133887-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-01-09 US disclosed
US-4127662-A ANTIACNE SCHERING CORPORATION (US) 1978-11-28 US disclosed
US-4123433-A ANTIACNE AGENTS SCHERING CORPORATION (US) 1978-10-31 US disclosed
US-4044140-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1977-08-23 US disclosed