SCHEMBL11534166

SCHEMBL11534166

Cc1ccc(C(c2ccccc2)(c2ccccc2)c2ccc(Br)nc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.38
ALDH1A1 P00352 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KIF11 P52732 9/20 0.37
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
LMNA P02545 1/20 0.33
ALOX12 P18054 1/20 0.33
ACHE P22303 1/20 0.33
CYP19A1 P11511 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11534894 0.91 NPC1 (0.33) TSHRALDH1A1SMN1; SMN2CYP19A1
SCHEMBL11533455 0.84 NPC1 (0.44) ALDH1A1SMN1; SMN2KIF11MEN1KMT2A
SCHEMBL11535231 0.83 KCNN4 (0.39) KIF11MEN1KMT2ACYP19A1
SCHEMBL11535711 0.83 CYP19A1 (0.40) TSHRSMN1; SMN2KIF11MEN1KMT2A
SCHEMBL11541379 0.83 ALDH1A1 (0.48) TSHRALDH1A1KIF11KMT2ALMNA
SCHEMBL11537892 0.82 KIF11 (0.41) ALDH1A1SMN1; SMN2KIF11MEN1KMT2A
SCHEMBL11533304 0.80 KIF11 (0.38) TSHRALDH1A1SMN1; SMN2KIF11MEN1
SCHEMBL8671538 0.79 TSHR (0.57) TSHRALDH1A1KIF11MEN1KMT2A
SCHEMBL9632111 0.79 TSHR (0.57) TSHRALDH1A1KIF11MEN1KMT2A
SCHEMBL14276997 0.79 TSHR (0.57) TSHRALDH1A1KIF11MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139625-A 5-(Substituted triphenylmethyl)picolinamides and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-13 US disclosed
US-4133887-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-01-09 US disclosed
US-4127662-A ANTIACNE SCHERING CORPORATION (US) 1978-11-28 US disclosed
US-4123433-A ANTIACNE AGENTS SCHERING CORPORATION (US) 1978-10-31 US disclosed
US-4044140-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1977-08-23 US disclosed