SCHEMBL11535231

SCHEMBL11535231

Fc1ccc(C(c2ccccc2)(c2ccc(F)cc2)c2ccc(Br)nc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 5/20 0.39
CYP19A1 P11511 3/20 0.36
TDP1 Q9NUW8 3/20 0.35
KIF11 P52732 3/20 0.34
GPR55 Q9Y2T6 1/20 0.34
KCNE1 P15382 1/20 0.33
KCNQ1 P51787 1/20 0.33
MLNR O43193 1/20 0.33
NR1I2 O75469 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
TBXA2R P21731 1/20 0.33
CCKBR P32239 1/20 0.33
OPRK1 P41145 1/20 0.33
SLC6A3 Q01959 1/20 0.33
KCNH2 Q12809 1/20 0.33
NR1H4 Q96RI1 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.31
USP2 O75604 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11534894 0.91 NPC1 (0.33) KCNN4CYP19A1RAB9A
SCHEMBL11537554 0.89 KCNN4 (0.40) KCNN4CYP19A1TDP1KIF11
SCHEMBL11541379 0.86 ALDH1A1 (0.48) CYP19A1TDP1KIF11KMT2ARAB9A
SCHEMBL11533455 0.84 NPC1 (0.44) CYP19A1KIF11MEN1KMT2ARAB9A
SCHEMBL11534166 0.83 TSHR (0.38) CYP19A1KIF11MEN1KMT2A
SCHEMBL11536103 0.83 CYP19A1 (0.42) KCNN4CYP19A1TDP1KIF11KMT2A
SCHEMBL11535711 0.83 CYP19A1 (0.40) CYP19A1KIF11MEN1KMT2ARAB9A
SCHEMBL11538690 0.82 KCNN4 (0.37) KCNN4KIF11KCNE1KCNQ1MLNR
SCHEMBL11533304 0.80 KIF11 (0.38) TDP1KIF11MEN1KMT2ARAB9A
SCHEMBL11535122 0.79 ALDH1A1 (0.35) CYP19A1TDP1KIF11KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4139625-A 5-(Substituted triphenylmethyl)picolinamides and their use as anti-acne agents SCHERING CORPORATION (US) 1979-02-13 US disclosed
US-4133887-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1979-01-09 US disclosed
US-4127662-A ANTIACNE SCHERING CORPORATION (US) 1978-11-28 US disclosed
US-4123433-A ANTIACNE AGENTS SCHERING CORPORATION (US) 1978-10-31 US disclosed
US-4044140-A Trityl picolinic acid derivatives and their use as anti-acne agents SCHERING CORPORATION (US) 1977-08-23 US disclosed